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Perkin Transactions 1 1972-2002 logo

Year 1996
Main Index

Issue 1


Front cover

pg X001; DOI:
10.1039/P199600FX001
PDF
Contents pages

pg P001; DOI:
10.1039/P199600FP001
PDF
Auxiliary accelerated reactions: catalytic hydrogenation
Andrew D. Westwell and Jonathan M. J. Williams
pg 1; DOI:
10.1039/P19960000001
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Novel approach to the synthesis of -alkoxycarbonyl -aminophosphonic esters based on a facile transformation of phosphoranes to phosphonic esters
Masahiko Seki Kazuhiko Kondo and Tameo Iwasaki
pg 3; DOI:
10.1039/P19960000003
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Back cover

pg X003; DOI:
10.1039/P199600BX003
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Cascade radical mediated macrocyclisation-transannulation reactions leading to ring-fused bicycles
Gerald Pattenden Allison J. Smithies David Tapolczay and Daryl S. Walter
pg 7; DOI:
10.1039/P19960000007
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Back matter

pg P007; DOI:
10.1039/P199600BP007
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A cascade radical macrocyclisation–transannulation approach towards the construction of ring-fused tricycles and polycycles
Michael J. Begley Gerald Pattenden Allison Smithies David Tapolczay and Daryl S. Walter
pg 21; DOI:
10.1039/P19960000021
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Consecutive 6-endo trigonal cyclisations from polyene acyl radical intermediates leading to decalone and perhydrophenanthrone ring constructions
Ligong Chen G. Bryon Gill Gerald Pattenden and Houri Simonian
pg 31; DOI:
10.1039/P19960000031
PDF
Acyl radical-mediated polyene cyclisations directed towards steroid ring synthesis
Andrei Batsanov Ligong Chen G. Bryon Gill and Gerald Pattenden
pg 45; DOI:
10.1039/P19960000045
PDF
Concise syntheses of cembrenes based on radical-mediated vinylcyclopropane ring-opening reactions in casbene
Gerald Pattenden and Allison J. Smithies
pg 57; DOI:
10.1039/P19960000057
PDF
Synthesis and solubility properties of C60 fullerene derivatives bearing carboxy groups
Hideo Tomioka and Katsutoshi Yamamoto
pg 63; DOI:
10.1039/P19960000063
PDF
Dioxygenase-catalysed oxidation of dihydronaphthalenes to yield arene hydrate and cis-dihydro naphthalenediols
Derek R. Boyd Narain D. Sharma Nuala A. Kerley R. Austin S. McMordie Gary N. Sheldrake Paul Williams and Howard Dalton
pg 67; DOI:
10.1039/P19960000067
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Preparation of some new intercalating europium(III) sensitizers
Stephen T. Mullins Peter G. Sammes Richard M. West and Gokhan Yahioglu
pg 75; DOI:
10.1039/P19960000075
PDF
Antitumour benzothiazoles. Part 2. Formation of 2,2-diaminobiphenyls from the decomposition of 2-(4-azidophenyl)benzazoles in trifluoromethanesulfonic acid
Malcolm F. G. Stevens Dong-Fang Shi and Angeles Castro
pg 83; DOI:
10.1039/P19960000083
PDF
Recoverable chiral sulfoxides for asymmetric synthesis: application to stereoselective carbonyl reduction and the asymmetric synthesis of allylic alcohols
Roger J. Butlin Ian D. Linney Mary F. Mahon Heather Tye and Martin Wills
pg 95; DOI:
10.1039/P19960000095
PDF
A study on the scope of the photochemical 1,3-migration of oximino groups in ,-unsaturated oximes and oxime derivatives
Diego Armesto Mar G. Gallego William M. Horspool and Ana Ramos
pg 107; DOI:
10.1039/P19960000107
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Instructions for authors (1996)

pg ixa; DOI:
10.1039/P19960000ixa
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Editorial

pg viia; DOI:
10.1039/P1996000viia
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Refereeing procedure and policy

pg xxxi; DOI:
10.1039/P1996000xxxi
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Conference diary

pg xxxv; DOI:
10.1039/P1996000xxxv
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Issue 2


Front cover

pg X005; DOI:
10.1039/P199600FX005
PDF
Back cover

pg X007; DOI:
10.1039/P199600BX007
PDF
Contents pages

pg P011; DOI:
10.1039/P199600FP011
PDF
Back matter

pg P017; DOI:
10.1039/P199600BP017
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Self-regulated molecular rearrangement: diastereoselective zwitterionic aza-Claisen protocol
Chan-Mo Yu Ha-Soon Choi Jongho Lee Won-Hyuk Jung and Hyuk-Jun Kim
pg 115; DOI:
10.1039/P19960000115
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Ring-opening reactions of pyrrolidinylcyclopropenyl cations in alkaline aqueous solution
Yoshio Yagyu Noboru Matsumura Hirokazu Tanaka Zyun Maeda and Hiroo Inoue
pg 117; DOI:
10.1039/P19960000117
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Stereoselective reaction of arylsulfanyl-stabilized homoenolates with aldehydes
Tsuyoshi Shinozuka Yuusuke Kikori Morio Asaoka and Hisashi Takei
pg 119; DOI:
10.1039/P19960000119
PDF
Rearrangement and radical mediated decarboxylation of trimethylsilyl benzoates using xenon difluoride
Pakawan Nongkunsarn and Christopher A. Ramsden
pg 121; DOI:
10.1039/P19960000121
PDF
New methodology for the synthesis of unsaturated 8-, 9- and 10-membered lactams
P. Andrew Evans Andrew B. Holmes Ross P. McGeary Alan Nadin Keith Russell Peter J. O'Hanlon and Neil D. Pearson
pg 123; DOI:
10.1039/P19960000123
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Detection of 2-substituted cyclobutanones as irradiation products of lipid-containing foods: synthesis and applications of cis- and trans-2-(tetradec-5-enyl)cyclobutanones and 11-(2-oxocyclobutyl)undecanoic acid
Lynne Hamilton M. Hilary Stevenson Derek R. Boyd Ian N. Brannigan Alan B. Treacy John T. G. Hamilton W. Colin McRoberts and Christopher T. Elliott
pg 139; DOI:
10.1039/P19960000139
PDF
A one-step photocatalytic synthesis of 2-(trifluoromethyl)butyrolactones
Ninja Reineke Naveed A. Zaidi Manju Mitra David O'Hagan Andrei S. Batsanov Judith A. K. Howard and Dmitri Y. Naumov
pg 147; DOI:
10.1039/P19960000147
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Asymmetric total synthesis of (–)-podophyllotoxin
Edward J. Bush and David W. Jones
pg 151; DOI:
10.1039/P19960000151
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Aziridination of alkenes using 3-acetoxyamino-2-trifluoromethylquinazolin-4(3H)-one
Robert S. Atkinson Michael P. Coogan and Clive L. Cornell
pg 157; DOI:
10.1039/P19960000157
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Synthetic studies on 4,5-dihydro-3H-1,2,4-triazole-3,5-diones bearing fluorogenic residues at N-4
Gordon Read and Nigel R. Richardson
pg 167; DOI:
10.1039/P19960000167
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On-resin solid-phase synthesis of asparagine N-linked glycopeptides: use of N-(2-acetoxy-4-methoxybenzyl)(AcHmb) aspartyl amide-bond protection to prevent unwanted aspartimide formation
John Offer Martin Quibell and Tony Johnson
pg 175; DOI:
10.1039/P19960000175
PDF
Synthesis and optical resolution of axially dissymmetric pyrroles and pyrocolls: new catalysts for the enantioselective addition of diethylzinc to aromatic aldehydes
Yoshio Furusho Akihiro Tsunoda and Takuzo Aida
pg 183; DOI:
10.1039/P19960000183
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Organozinc reagents in synthesis: the facile generation of 2-(trialkylsilyl)prop-2-enylzinc from 2-bromo-1-trimethylsilylprop-2-ene
James J. Eshelby Philip J. Parsons and Patrick J. Crowley
pg 191; DOI:
10.1039/P19960000191
PDF
Tetracyclic triterpenes. Part 16. Synthesis of 31-norcucurbitane and fusidane derivatives in the skeletal rearrangements of 9,11-epoxy-4-demethyl-5-lanostanes
Zdzisaw Paryzek and Jacek Martynow
pg 201; DOI:
10.1039/P19960000201
PDF
An asymmetric total synthesis of (+)-(3R,4S,5R,7S)-neoclausenamide
Jian-qiang Wang and Wei-sheng Tian
pg 209; DOI:
10.1039/P19960000209
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Studies on Rubia akane(RA) derivatives. Part 8. Design, syntheses and antitumour activity of cyclic hexapeptide RA analogues possessing an alkyl substituent on the Tyr-3 aromatic ring
Yukio Hitotsuyanagi Suguru Lee Izumi Ito Kazuyuki Kondo Koichi Takeya Takehiro Yamagishi Takatoshi Nagate and Hideji Itokawa
pg 213; DOI:
10.1039/P19960000213
PDF
Stereoselectivity in the photoinduced electron transfer (PET) promoted intramolecular cyclisations of 1-alkenyl-2-silyl-piperidines and -pyrrolidines: rapid construction of 1-azabicyclo[m.n.0]alkanes and stereoselective synthesis of ()-isoretronecanol and ()-epilupinine
Ganesh Pandey Gottimukkula Devi Reddy and Debasish Chakrabarti
pg 219; DOI:
10.1039/P19960000219
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Conference diary

pg viib; DOI:
10.1039/P1996000viib
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Issue 3


Front cover

pg X009; DOI:
10.1039/P199600FX009
PDF
Back cover

pg X011; DOI:
10.1039/P199600BX011
PDF
Contents pages

pg P021; DOI:
10.1039/P199600FP021
PDF
Back matter

pg P025; DOI:
10.1039/P199600BP025
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Synthesis of fused 1,2,4-thiadiazoles from -amino nitriles and thioacyl isothiocyanates
Gerrit L'abbé Bart D'hooge and Wim Dehaen
pg 225; DOI:
10.1039/P19960000225
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Convenient synthesis of enantiopure cyclic -hydroxyalkyl -amino esters
Mark D. Andrews Andrew G. Brewster Mark G. Moloney and Karen L. Owen
pg 227; DOI:
10.1039/P19960000227
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Studies on isocyanides and related compounds: synthesis of benzo[c]thiophenes by way of acid-induced three-component reactions
Ricardo Bossio Stefano Marcaccini Roberto Pepino and Tomás Torroba
pg 229; DOI:
10.1039/P19960000229
PDF
Generation of 6-alkylidene/benzylidene-3,6-dihydropyrazin-2(1H)ones by reaction of 6-bromomethylpyrazin-2(1H)-ones with methoxide and further conversion into specific piperazine-2,5-diones and pyrazin-2(1H)-ones
Kris J. Buysens Didier M. Vandenberghe Suzanne M. Toppet and Georges J. Hoornaert
pg 231; DOI:
10.1039/P19960000231
PDF
Penochalasins, a novel class of cytotoxic cytochalasans from a Penicillium species separated from a marine alga: structure determination and solution conformation
Atsushi Numata Chika Takahashi Yoshinori Ito Katsuhiko Minoura Takeshi Yamada Chitose Matsuda and Kyosuke Nomoto
pg 239; DOI:
10.1039/P19960000239
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Methyl 3-(triphenylphosphoranylideneamino)pyrazine-2-carboxylate: synthesis, crystal structure and use in pteridin-4(3H)ones synthesis
Tomohiro Okawa Shoji Eguchi and Akikazu Kakehi
pg 247; DOI:
10.1039/P19960000247
PDF
Chemoenzymatic synthesis of carbocyclic nucleoside analogues with bicyclo[3.1.0]hexyl residues
Fritz Theil Sibylle Ballschuh Martin von Janta-Lipinski and Roger A. Johnson
pg 255; DOI:
10.1039/P19960000255
PDF
Transformations of isoxazolidine and dihydropyran derivatives to optically active compounds
Angel Díaz-Ortiz Enrique Díez-Barra Antonio de la Hoz Pilar Prieto and Andrés Moreno
pg 259; DOI:
10.1039/P19960000259
PDF
Preparation of secondary amines by reductive amination with metallic magnesium
Ivan V. Miovi M. D. Ivanovi Goran M. Rogli Vesna D. Kiricojevi and Jelena B. Popovi
pg 265; DOI:
10.1039/P19960000265
PDF
Decomposition of 2-dialkylaminobenzoyl azides to yield isocyanates and 1,1-dialkylindazol-1-ium-3-olates
Norman M. Waldron and Muhammad Raza
pg 271; DOI:
10.1039/P19960000271
PDF
Synthesis and inclusion properties of pyridinophane-linked macrocycles
Hiroyuki Takemura Satoshi Osada Teruo Shinmyozu and Takahiko Inazu
pg 277; DOI:
10.1039/P19960000277
PDF
Photocyclisation of enamides. Part 39. General strategy for the synthesis of pseudodistomins: synthesis of triacetates of ()-tetrahydropseudodistomin and proposed structures of pseudodistomins A and B
Takeaki Naito Yoko Yuumoto Toshiko Kiguchi and Ichiya Ninomiya
pg 281; DOI:
10.1039/P19960000281
PDF
Convenient procedure for converting 1,3-dithiolane-2-thiones into 1,3-dithiolan-2-ones
Margherita Barbero Iacopo Degani Stefano Dughera Rita Fochi and Laura Piscopo
pg 289; DOI:
10.1039/P19960000289
PDF
Improved synthesis of brassinolide
Trevor C. McMorris Rodrigo G. Chavez and Prakash A. Patil
pg 295; DOI:
10.1039/P19960000295
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Conference diary

pg v; DOI:
10.1039/P1996000000v
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Issue 4


Front cover

pg X013; DOI:
10.1039/P199600FX013
PDF
Back cover

pg X015; DOI:
10.1039/P199600BX015
PDF
Contents pages

pg P029; DOI:
10.1039/P199600FP029
PDF
Back matter

pg P035; DOI:
10.1039/P199600BP035
PDF
Synthetic studies towards pseudopterosin A
Lars Eklund Ian Sarvary and Torbjörn Frejd
pg 303; DOI:
10.1039/P19960000303
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Synthesis of dendritic polypyridines with ethoxycarbonyl groups as surface functionality
Gavino Chessa and Alberto Scrivanti
pg 307; DOI:
10.1039/P19960000307
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The potential of sulfimides as chiral acyl anion equivalents
Gareth Smith Tim J. Sparey and Paul C. Taylor
pg 313; DOI:
10.1039/P19960000313
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Photoinduced skeletal rearrangement of 1,1-diarylspiropentanes
Yasutake Takahashi Hitoshi Ohaku Shin-ichi Morishima Takanori Suzuki Hiroshi Ikeda and Tsutomu Miyashi
pg 319; DOI:
10.1039/P19960000319
PDF
Reactions of -trimethylsilylvinyl carbanions with carboxylic acid derivatives: the relationship between product distribution and substrate reactivity
Alan R. Bassindale Ibrahim Katampe Patricia A. Kyle and Peter G. Taylor
pg 327; DOI:
10.1039/P19960000327
PDF
Diastereoselective conversion of sulfides into sulfoxides. 1,5- and 1,6-asymmetric induction
Justin F. Bower Christopher J. Martin David J. Rawson Alexandra M. Z. Slawin and Jonathan M. J. Williams
pg 333; DOI:
10.1039/P19960000333
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Development of the juli asymmetric epoxidation reaction. Part 1. Application of the oxidation to enones other than chalcones
M. Elena Lasterra-Sánchez Ulfried Felfer Patrick Mayon Stanley M. Roberts Steven R. Thornton and Christine J. Todd
pg 343; DOI:
10.1039/P19960000343
PDF
Synthesis of C-D-ring analogues of the azasteroid A25822
Andrew J. Sutherland James K. Sutherland and Patrick J. Crowley
pg 349; DOI:
10.1039/P19960000349
PDF
Novel reductase participation in the syn-addition of hydrogen to the CC bond of enones in the cultured cells of Nicotiana tabacum
Kei Shimoda Diana I. Ito Shunsuke Izumi and Toshifumi Hirata
pg 355; DOI:
10.1039/P19960000355
PDF
Stereocontrolled synthesis of E-homoallylic sulfides with 1,4,5 related chiral centres using the [2,3] sigmatropic rearrangement of sulfonium ylides
Richard C. Hartley Ian C. Richards and Stuart Warren
pg 359; DOI:
10.1039/P19960000359
PDF
Synthesis of nitrogen-containing unsaturated carbohydrates via an allyl cyanate-to-isocyanate rearrangement
Yoshiyasu Ichikawa Chie Kobayashi and Minoru Isobe
pg 377; DOI:
10.1039/P19960000377
PDF
Preparation and enantiomer recognition behaviour of azophenolic crown ethers containing cis-1-phenylcyclohexane-l,2-diol as the chiral subunit and 2,4-dinitrophenylazophenol as the chromophore
Koichiro Naemura Koji Ueno Sachiko Takeuchi Keiji Hirose Yoshito Tobe Takahiro Kaneda and Yoshiteru Sakata
pg 383; DOI:
10.1039/P19960000383
PDF
Stereocontrol in radical-mediated allylation of acyclic -bromo--siloxy esters by complexation with lanthanide shift reagents Ln(fod)3
Hajime Nagano Yukie Kuno Yuriko Omori and Mayumi Iguchi
pg 389; DOI:
10.1039/P19960000389
PDF
Synthesis and stereochemistry of the epoxides of 2-arylmethylidene-1-tetralones
Waldemar Adam Judit Halász Zsigmond Jámbor Albert Lévai Csaba Nemes Tamás Patonay and Gábor Tóth
pg 395; DOI:
10.1039/P19960000395
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Conference diary

pg viic; DOI:
10.1039/P1996000viic
PDF

Issue 5


Front cover

pg X017; DOI:
10.1039/P199600FX017
PDF
Back cover

pg X019; DOI:
10.1039/P199600BX019
PDF
Contents pages

pg P037; DOI:
10.1039/P199600FP037
PDF
Back matter

pg P043; DOI:
10.1039/P199600BP043
PDF
Studies directed towards the synthesis of herbicidins. Model study based on late stage N-glycosylation
Hayley M. Binch and Timothy Gallagher
pg 401; DOI:
10.1039/P19960000401
PDF
Total synthesis of ()-methylenolactocin by radical cyclisation of an epoxide using a transition-metal radical
Gourhari Maiti and Subhas Chandra Roy
pg 403; DOI:
10.1039/P19960000403
PDF
Enantioselective total synthesis of the di-O-methyl ethers of (–)-agatharesinol, (+)-hinokiresinol and (–)-sugiresinol, characteristic norlignans of Coniferae
Osamu Muraoka Bao-Zhong Zheng Noriyuki Fujiwara and Genzoh Tanabe
pg 405; DOI:
10.1039/P19960000405
PDF
Selectivity in the ring-expansion and ring-switching reactions of bicyclooxonium ions

pg 413; DOI:
10.1039/P19960000413
PDF
A new synthesis of pyrroles and porphyrins fused with aromatic rings
Noboru Ono Hideo Hironaga Kazuo Ono Syunichi Kaneko Takashi Murashima Takahiro Ueda Chikanori Tsukamura and Takuji Ogawa
pg 417; DOI:
10.1039/P19960000417
PDF
Stereospecific formation of R-aromatic acyloins by Zymomonas mobilis pyruvate decarboxylase
Stephen Bornemann David H. G. Crout Howard Dalton Vladimír Kren Mario Lobell Gregory Dean Nicholas Thomson and Margaret M. Turner
pg 425; DOI:
10.1039/P19960000425
PDF
Synthesis of 2-deoxy-- and --D-arabino-hexopyranosyl phosphonic acids and related compounds; analogues of early intermediates in the shikimate pathway
Nigel J. Barnes Mark A. Probert and Richard H. Wightman
pg 431; DOI:
10.1039/P19960000431
PDF
Synthesis of C11 chain-extended analogues of N-acetylneuraminic acid
Milton J. Kiefel Simon Bennett and Mark von Itzstein
pg 439; DOI:
10.1039/P19960000439
PDF
Diels–Alder reactions of o-benzoquinones with acyclic dienes
Vijay Nair and Sasi Kumar
pg 443; DOI:
10.1039/P19960000443
PDF
An improved procedure for the synthesis of substituted acetylenes from the reaction of acetylene gas with aryl iodides under palladium–copper catalysis
Manojit Pal and Nitya G. Kundu
pg 449; DOI:
10.1039/P19960000449
PDF
Oxidative removal of 1,3-dithiane protecting groups by 2,3-dichloro-5,6-dicyano-p-benzoquinone (DDQ)
Kiyoshi Tanemura Hiroshi Dohya Masanori Imamura Tsuneo Suzuki and Takaaki Horaguchi
pg 453; DOI:
10.1039/P19960000453
PDF
Condensed heteroaromatic ring systems. Part 24. Synthesis of rigidin, a pyrrolo[2,3-d]pyrimidine marine alkaloid
Takao Sakamoto Yoshinori Kondo Shuichiroh Sato and Hiroshi Yamanaka
pg 459; DOI:
10.1039/P19960000459
PDF
Highly diastereoselective route to trans-5-substituted 2-hydroxymethylpyrrolidine derivatives by radical cyclisation
Yoko Yuasa Jun Ando and Shiroshi Shibuya
pg 465; DOI:
10.1039/P19960000465
PDF
Flash vacuum pyrolysis of stabilised phosphorus ylides. Part 7. Cyclisation of amino acid derived -phtnalimidoacyl ylides to give pyrroloisoindolediones
R. Alan Aitken Harris R. Cooper and Amit P. Mehrotra
pg 475; DOI:
10.1039/P19960000475
PDF
Flash vacuum pyrolysis of stabilised phosphorus ylides. Part 8. Preparation of symmetrical and unsymmetrical 1,3-diynes from alkynoyl ylides and oxalyl diylides
R. Alan Aitken Hugues Hérion Caroline E. R. Horsburgh Nazira Karodia and Shirley Seth
pg 485; DOI:
10.1039/P19960000485
PDF
Synthesis and study of 3-(triphenylphosphoranylidene)-2,3-dihydro-1H-indol-2-one
George E. Lathourakis and Konstantinos E. Litinas
pg 491; DOI:
10.1039/P19960000491
PDF
Conference diary

pg viid; DOI:
10.1039/P1996000viid
PDF

Issue 6


Front cover

pg X021; DOI:
10.1039/P199600FX021
PDF
Back cover

pg X023; DOI:
10.1039/P199600BX023
PDF
Contents pages

pg P049; DOI:
10.1039/P199600FP049
PDF
Back matter

pg P055; DOI:
10.1039/P199600BP055
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Oxocarbons and related compounds. Part 24. chlorosquarylation of indoles
Arthur H. Schmidt Stefan H. Thiel and Otfried Gaschler
pg 495; DOI:
10.1039/P19960000495
PDF
Oxocarbons and related compounds. Part 25. Heterocycle-fused benzocyclobutenediones. Synthesis of indolo-, benzofuro- and benzothieno-dihydrobenzocyclobutenediones and benzocyclobutenediones
Arthur H. Schmidt Kai O. Lechler Thorsten Pretz and Ingo Franz
pg 497; DOI:
10.1039/P19960000497
PDF
Cycloaddition of tetracyanoethene oxide with [60]fullerene
Nadine Jagerovic José Elguero and Jean-Louis Aubagnac
pg 499; DOI:
10.1039/P19960000499
PDF
Absence of the alleged retardation of the Diels–Alder reaction for dienes bearing a neighbouring hydroxy substituent
Paul Glossop and David W. Jones
pg 501; DOI:
10.1039/P19960000501
PDF
Stereospecific synthesis of (2S,4R)-[5,5,5-2H3]leucine
Ryan A. August Jeffrey A. Khan Claire M. Moody and Douglas W. Young
pg 507; DOI:
10.1039/P19960000507
PDF
A route to dihydro[2]benzooxepino[4,5-c]pyridines and dihydrothieno[d][2]benzooxepines via the 1.7-electrocyclisation of carbonyl ylides
Donal F. O'Shea and John T. Sharp
pg 515; DOI:
10.1039/P19960000515
PDF
Diels–Alder reactions of trichloro-1,2,4-triazine: intramolecular additions with 1,5 and 1,6 dienes
Michael G. Barlow Lakhdar Sibous Nadia N. E. Suliman and Anthony E. Tipping
pg 519; DOI:
10.1039/P19960000519
PDF
Enzymic synthesis of hemithiocellodextrins
Vincent Moreau and Hugues Driguez
pg 525; DOI:
10.1039/P19960000525
PDF
Inter- and intra-molecular selectivity in the cyclisation of N-cinnamoyl-1-naphthamides in solid-state photochemistry and peri selectivity in their photocyclisation in solution
Shigeo Kohmoto Takashi Kobayashi Takehiko Nishio Ikuo Iida Keiki Kishikawa Makoto Yamamoto and Kazutoshi Yamada
pg 529; DOI:
10.1039/P19960000529
PDF
Synthesis of enantiopure -deuteriated Boc-L-amino acids
Yiannis Elemes and Ulf Ragnarsson
pg 537; DOI:
10.1039/P19960000537
PDF
Synthesis and X-ray structure of 1,4-bis[4-(N,N-dimethylamino)phenyl]buta-1,3-diyne: charge-transfer complex with acceptors
J. Gonzalo Rodríguez Santiago Ramos Rosa Martín-Villamil Isabel Fonseca and Armando Albert
pg 541; DOI:
10.1039/P19960000541
PDF
Synthesis of 1-amino-1,2,3,14b-tetrahydro-4H-pyrido[1,2-d]-dibenzo[b,f][1,4]oxazepine and related compounds
Wilson L. Caulfield Samuel Gibson and Duncan R. Rae
pg 545; DOI:
10.1039/P19960000545
PDF
Reactions of carbene intermediates from the reaction of trialkyl phosphites with dialkyl benzoylphosphonates: intramolecular cyclisations of 2-substituted dialkyl benzoylphosphonates
D. Vaughan Griffiths Penelope A. Griffiths Khalku Karima and Belinda J. Whitehead
pg 555; DOI:
10.1039/P19960000555
PDF
Thermolysis and photolysis of 1-substituted triptycenes. Divergent fragmentation pathways of the triptycyl skeleton
Hideo Tomioka and Junichi Nakajima
pg 563; DOI:
10.1039/P19960000563
PDF
Potential intermediate, ()-di-o-acetyl-3-phenylselanyl-3,3a-dihydro-B-nor-6,7a-secolycorin-5-one for synthesis of the Amaryllidaceae alkaloid lycorine: formal and total syntheses of ()-lycorine
Osamu Hoshino Miyuki Ishizaki Keisuke Kamei Minoru Taguchi Takashi Nagao Kiyoshi Iwaoka Shohei Sawaki Bunsuke Umezawa and Yoichi Iitaka
pg 571; DOI:
10.1039/P19960000571
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Stereoselective synthesis of N-acetyl thiochitooligosaccharides. Different behaviours of methyl N-acetyl-- and --thiochitobiosides during acetolysis
Lai-Xi Wang and Yuan C. Lee
pg 581; DOI:
10.1039/P19960000581
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Conference diary

pg viie; DOI:
10.1039/P1996000viie
PDF

Issue 7


Front cover

pg X025; DOI:
10.1039/P199600FX025
PDF
Back cover

pg X027; DOI:
10.1039/P199600BX027
PDF
Contents pages

pg P057; DOI:
10.1039/P199600FP057
PDF
Back matter

pg P065; DOI:
10.1039/P199600BP065
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Asymmetric induction using novel chiral auxiliaries derived from D-glucose
Vijay Nair and Jaya Prabhakaran
pg 593; DOI:
10.1039/P19960000593
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First synthesis of -2-deoxy[9-15N]adenosine
Charles C. Orji Joe Kelly David A. Ashburn and Louis A. Silks III
pg 595; DOI:
10.1039/P19960000595
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Calixarene-bound dendritic macromolecules
George Ferguson John F. Gallagher M. Anthony McKervey and Evelyn Madigan
pg 599; DOI:
10.1039/P19960000599
PDF
New preparative method for optically active 2,2- and 4,4-dihydroxybiphenyl derivatives. A new chiral host compound 4,4-dihydroxy-2,2,3,3,6,6-hexamethylbiphenyl
Koichi Tanaka Ayao Moriyama and Fumio Toda
pg 603; DOI:
10.1039/P19960000603
PDF
Elemental fluorine. Part 1. Synthesis of fluoroaromatic compounds
Richard D. Chambers Christopher J. Skinner John Hutchinson and Julie Thomson
pg 605; DOI:
10.1039/P19960000605
PDF
Synthetic studies towards the clerodane insect antifeedant jodrellin A: preparation of a polycyclic model compound with antifeedant activity
Ana C. Cuñat David Díez-Martín Steven V. Ley and Francis J. Montgomery
pg 611; DOI:
10.1039/P19960000611
PDF
Enantioselective synthesis of 2-substituted 4-aminobutanoic acid (GABA) analogues via cyanomethylation of chiral enolates
Shamim Azam Alice A. D'Souza and Peter B. Wyatt
pg 621; DOI:
10.1039/P19960000621
PDF
Reinvestigation of reactions of thiazolium and benzothiazolium N-phenacylides with electron-deficient acetylenes
Tatsunori Iwamura Masahiro Kobayashi Takashi Ichikawa Hiroshi Shimizu and Tadashi Kataoka
pg 629; DOI:
10.1039/P19960000629
PDF
Enantioselective synthesis of the 13-membered macrodiolide bartanol
John A. O'Neill Stephen D. Lindell Thomas J. Simpson and Christine L. Willis
pg 637; DOI:
10.1039/P19960000637
PDF
Synthesis and effects on arginase and nitric oxide synthase of two novel analogues of N-hydroxyarginine, N-hydroxyindospicine and p-hydroxyamidinophenylalanine
Sandrine Vadon Julien Custot Jean-Luc Boucher and Daniel Mansuy
pg 645; DOI:
10.1039/P19960000645
PDF
Synthesis of polyester dendrimers
David M. Haddleton Hardeep S. Sahota Paul C. Taylor and Stephen G. Yeates
pg 649; DOI:
10.1039/P19960000649
PDF
1,5-Diborabicyclo[3.3.3]undecane; thermolysis of the product from hydroboration of triallylborane with triethylamine–borane
Roger W. Alder and Zhao Jin
pg 657; DOI:
10.1039/P19960000657
PDF
The generation and synthetic applications of episulfone -anions
Andrew E. Graham Wendy A. Loughlin Madeleine H. Moore Simon M. Pyke Giles Wilson and Richard J. K. Taylor
pg 661; DOI:
10.1039/P19960000661
PDF
Photolysis of fluorodiphenylamines
Paul W. Groundwater David Hughes Michael B. Hursthouse and Rhiannon Lewis
pg 669; DOI:
10.1039/P19960000669
PDF
Intramolecular radical substitution reactions: a novel approach to fused [1,2-a] indoles
Stephen Caddick Karim Aboutayab Kerry Jenkins and Robert I. West
pg 675; DOI:
10.1039/P19960000675
PDF
Synthesis of (2S)-O-phosphohomoserine and its C-2 deuteriated and C-3 chirally deuteriated isotopomers: probes for the pyridoxal phosphate-dependent threonine synthase reaction
Fiona Barclay Ewan Chrystal and David Gani
pg 683; DOI:
10.1039/P19960000683
PDF
Asymmetric synthesis of amines using a chiral, non-racemic, benzylidene sulfinamide derived from a recoverable precursor
David R. J. Hose Mary F. Mahon Kieran C. Molloy Tony Raynham and Martin Wills
pg 691; DOI:
10.1039/P19960000691
PDF
Intramolecular Diels–Alder additions to 2-benzopyran-3-ones; endo-selective additions and some reactions of the adducts
David W. Jones and Firstborn Matthew Nongrum
pg 705; DOI:
10.1039/P19960000705
PDF
Synthesis of the key component for preparation of 6-ketoprostaglandins by a two-component coupling process: synthesis of 6-keto-prostaglandin E1, ornoprostil and 2-trans-6-ketoprostaglandin E1
Yasufumi Kawanaka Naoya Ono Yukio Yoshida Sentaro Okamoto and Fumie Sato
pg 715; DOI:
10.1039/P19960000715
PDF
Backbone protection and its application to the synthesis of a difficult phosphopeptide sequence
Tony Johnson Leonard C. Packman Carolyn B. Hyde David Owen and Martin Quibell
pg 719; DOI:
10.1039/P19960000719
PDF
Synthesis of 2-allyl-2,3-dihydro-1H-indol-3-ones using in situ Claisen rearrangement of 2,3-dihydro-1H-indol-3-ones with allyl alcohols
Tomomi Kawasaki Kouhei Masuda Yasutaka Baba Romi Terashima Kana Takada and Masanori Sakamoto
pg 729; DOI:
10.1039/P19960000729
PDF
Structure of new anthocyanin-derived wine pigments
Hélène Fulcrand Paulo-Jorge Cameira dos Santos Pascale Sarni-Manchado Véronique Cheynier and Jean Favre-Bonvin
pg 735; DOI:
10.1039/P19960000735
PDF
Synthesis and characterization of bis[1.1.1]orthocyclophano-18-crown-6 compounds
Hiroshi Hara Shin-ichi Watanabe Makoto Yamada and Osamu Hoshino
pg 741; DOI:
10.1039/P19960000741
PDF
Base-induced cycloreversion of nitrile oxide cycloadducts: conversion of imines into secondary and tertiary amides and aromatic aldehydes into acids without a conventional oxidising agent
R. Alan Aitken and Swati V. Raut
pg 747; DOI:
10.1039/P19960000747
PDF
Conference diary

pg ixb; DOI:
10.1039/P19960000ixb
PDF

Issue 8


Front cover

pg X029; DOI:
10.1039/P199600FX029
PDF
Back cover

pg X031; DOI:
10.1039/P199600BX031
PDF
Contents pages

pg P067; DOI:
10.1039/P199600FP067
PDF
Back matter

pg P073; DOI:
10.1039/P199600BP073
PDF
Synthesis of N-2-adamantyloxymethylhistidine, his(N-2-adom), and its evaluation for peptide synthesis
Yoshio Okada Jidong Wang Takeshi Yamamoto and Yu Mu
pg 753; DOI:
10.1039/P19960000753
PDF
Designer yeast: a new reagent for enantioselective Baeyer–Villiger oxidations
Jon D. Stewart Kieth W. Reed and Margaret M. Kayser
pg 755; DOI:
10.1039/P19960000755
PDF
A highly asymmetric, Lewis acid-catalysed Diels–Alder reaction using optically active 2-(3-tolyl p-sulfinyl)furyl ,-unsaturated ketones as a dienophile
Yoshitsugu Arai Tsutomu Masuda Yukio Masaki and Motoo Shiro
pg 759; DOI:
10.1039/P19960000759
PDF
Palladium-catalysed arylation and alkenylation of cis-trifluoroprop-1-enyl methyl ether. A novel entry into trifluoromethylated compounds
Guo-qiang Shi Xian-hai Huang and Feng Hong
pg 763; DOI:
10.1039/P19960000763
PDF
Stereoselective synthesis of (E)-vinylic selenides via hydrozirconation of alk-1-ynes
Xian Huang and Liu-Sheng Zhu
pg 767; DOI:
10.1039/P19960000767
PDF
Radical addition to carbenoids. Chain reactions of -diazo carbonyl compounds with triorganotin hydrides, tris(trimethylsilyl)silane and allyltributylstannane
Hai-Shan Dang and Brian P. Roberts
pg 769; DOI:
10.1039/P19960000769
PDF
Product diversity in cyclisations of maleamic acids: the imide–isoimide dichotomy
John E. T. Corrie Madeleine H. Moore and Giles D. Wilson
pg 777; DOI:
10.1039/P19960000777
PDF
Preparation and chemistry of new unsymmetrically substituted tetrachalcogenofulvalenes bearing CN(CH2)2X and HO(CH2)2X groups (X = S or Se)
Laurent Binet Jean Marc Fabre Claude Montginoul Klaus Baek Simonsen and Jan Becher
pg 783; DOI:
10.1039/P19960000783
PDF
Photochemical reactions of 1-naphthylamines and haloforms: formation of bis(4-amino-1-naphthyl)methylium salts with remarkably long-wave electronic absorption
Koko Maeda Yumiko Horikoshi Mariko Hayashi Yukie Mori and Hajime Nagano
pg 789; DOI:
10.1039/P19960000789
PDF
Diastereoselective synthesis of 2,5-disubstituted 3-hydroxypyrrolidine and 2,6-disubstituted 3-hydroxypiperidine derivatives by radical cyclisation; synthesis of (+)-bulgecinine and (–)-desoxoprosopinine
Yoko Yuasa Jun Ando and Shiroshi Shibuya
pg 793; DOI:
10.1039/P19960000793
PDF
Preparation of optically active 3-substituted piperidines via ring expansion: synthesis of 4-amino- and 4-fluoro-1,4,5-trideoxy-1,5-imino-D-ribitol and 1,5-dideoxy-1,5-imino-D-ribitol
Dae-Kee Kim Ganghyeok Kim and Young-Woo Kim
pg 803; DOI:
10.1039/P19960000803
PDF
Some diphenylphosphorus(V) group monosaccharide compounds derived from methyl 2,3-O-isopropylidene--D-mannofuranoside
Martyn A. Brown Philip J. Cox R. Alan Howie Olga A. Melvin and James L. Wardell
pg 809; DOI:
10.1039/P19960000809
PDF
Co-cyclizations of nitrogen-containing acetylenes induced by a nickel triphenylphosphine complex to give aminoindane, isoindoline and isoindolinone derivatives
D. Malcolm Duckworth Simon Lee-Wong Alexandra M. Z. Slawin Edward H. Smith and David J. Williams
pg 815; DOI:
10.1039/P19960000815
PDF
Efficient stereocontrolled synthesis of D-erythro-sphingosine from N-benzoyl-D-glucosamine
Teiichi Murakami and Masakatsu Hato
pg 823; DOI:
10.1039/P19960000823
PDF
Formal total synthesis of trichodiene via skeletal rearrangement of regioselective photochemical [2 + 2] cycloadducts from cyclohexene derivatives
Yoshikazu Kitano Junko Fukuda Kazuhiro Chiba and Masahiro Tada
pg 829; DOI:
10.1039/P19960000829
PDF
v-Triazolines. Part 36. New synthesis of ethyl 1-alkyl-1,4,5,6-tetrahydro-6-oxopyridine-3-carboxylates and 1-alkyl-1,4,5,6-tetranydro-6-oxopyridine-3-carbonitriles through reduction of N-2-nitroarylamidines
Roberto Angelini Emanuela Erba and Donato Pocar
pg 837; DOI:
10.1039/P19960000837
PDF
Total synthesis of 3-hydroxy-6-oxaestra-1,3,5(10)-trien-17-one
Zhisong Cao and Joachim G. Liehr
pg 841; DOI:
10.1039/P19960000841
PDF
Taxol and taxane formation in plant cell culture
Peter Heinstein Jin-yun Zhou Mansi Wang Yeuk-Chuen Liu Xiao-ya Chen Dian Chen Steven H. Hoke II R. Graham Cooks and Ching-jer Chang
pg 845; DOI:
10.1039/P19960000845
PDF
Dolastatins 23: stereospecific synthesis of dolaisoleuine
George R. Pettit Douglas D. Burkett and Michael D. Williams
pg 853; DOI:
10.1039/P19960000853
PDF
Dolastatins 24: synthesis of (–)-dolastatin 10. X-Ray molecular structure of N,N-dimethylvalyl-valyl-dolaisoleuine tert-butyl ester
George R. Pettit Jayaram K. Srirangam Sheo Bux Singh Michael D. Williams Delbert L. Herald József Barkóczy Darko Kantoci and Fiona Hogan
pg 859; DOI:
10.1039/P19960000859
PDF
Conference diary

pg viif; DOI:
10.1039/P1996000viif
PDF

Issue 9


Front cover

pg X033; DOI:
10.1039/P199600FX033
PDF
Back cover

pg X035; DOI:
10.1039/P199600BX035
PDF
Front matter

pg P077; DOI:
10.1039/P199600FP077
PDF
Back matter

pg P083; DOI:
10.1039/P199600BP083
PDF
Simple one-pot transformations of toluene-p-sulfonates of 2,3-epoxy alcohols into allylic alcohols
Nobutaka Fujii Hiromu Habashita Masako Akaji Kazuo Nakai Toshiro Ibuka Masahiro Fujiwara Hirokazu Tamamura and Yoshinori Yamamoto
pg 865; DOI:
10.1039/P19960000865
PDF
Facile preparation of vinylaziridines by the reaction of N-sulfonylimines and cinnamyl bromide mediated by a catalytic amount of dimethyl sulfide
An-Hu Li Li-Xin Dai and Xue-Long Hou
pg 867; DOI:
10.1039/P19960000867
PDF
Synthesis and reaction of cyano-substitued 1,2,4-trioxolanes
Hajime Kuwabara Yoshihiro Ushigoe and Masatomo Nojima
pg 871; DOI:
10.1039/P19960000871
PDF
Diastereoselective addition of allylmetal compounds to imines derived from (S)-1-phenylethanamine
Giuseppe Alvaro Carla Boga Diego Savoia and Achille Umani-Ronchi
pg 875; DOI:
10.1039/P19960000875
PDF
Synthesis of 1-acylamino-1-(trimethylsiloxy)alkanes by trimethylsilyl trifluoromethanesulfonate-catalysed addition of bis(trimethylsilyl)amides to aldehydes
A. Peter Johnson Richard W. A. Luke Robert W. Steele and Andrew N. Boa
pg 883; DOI:
10.1039/P19960000883
PDF
Reactions of 1-acylamino-1-(trimethylsiloxy)alkanes: versatile precursors to acylimines
A. Peter Johnson Richard W. A. Luke and Andrew N. Boa
pg 895; DOI:
10.1039/P19960000895
PDF
Synthesis and reactions of N,N-bis[1-(trimethylsiloxy)alkyl]-formamides: preparation of ()-argemonine and ()-norargemonine
A. Peter Johnson Richard W. A. Luke Gurmaj Singh and Andrew N. Boa
pg 907; DOI:
10.1039/P19960000907
PDF
Facile conversion of perfluoroacyl fluorides into other acyl halides
Haruhiko Fukaya Tomonori Matsumoto Eiji Hayashi Yoshio Hayakawa and Takashi Abe
pg 915; DOI:
10.1039/P19960000915
PDF
Photoaddition of benzoxazole-2-thiones with alkenes
Takehiko Nishio Yo-ichi Mori Ikuo Iida and Akira Hosomi
pg 921; DOI:
10.1039/P19960000921
PDF
Strong solid base reagents and catalysts based on carbonaceous supports
Russell S. Drago and Krzysztof Jurczyk
pg 927; DOI:
10.1039/P19960000927
PDF
Reaction of in-situ generated -silylated allylic phosphonate carbanions with aldehydes. An unexpected cyclization reaction
Hashim Al-Badri Elie About-Jaudet and Noël Collignon
pg 931; DOI:
10.1039/P19960000931
PDF
Cyclo(-arginyl-sarcosyl-aspartyl-phenylglycyl-)2. Simple synthesis of an RGD-related peptide with inhibitory activity for platelet aggregation
Norikazu Nishino Jun Hayashida Toru Arai Hisakazu Mihara Yukio Ueno and Hiromichi Kumagai
pg 939; DOI:
10.1039/P19960000939
PDF
Synthesis of methyl 4-aryl-6-methyl-4,7-dihydro-1H-pyrazolo-[3,4-b]pyridine-5-carboxylates from methyl 4-aryl-6-methyl-2-oxo-1,2,3,4-tetrahydropyridine-5-carboxylates
Yamila Verdecia Margarita Suárez Alhmed Morales Elena Rodríguez Estael Ochoa Leandro González Nazario Martín Margarita Quinteiro Carlos Seoane and José L. Soto
pg 947; DOI:
10.1039/P19960000947
PDF
Syntheses of crown ether-esters with (benzyloxy)methyl side arms using SbPh3 and BiPh3 as templates1
Yoichi Habata Fumio Fujishiro and Sadatoshi Akabori
pg 953; DOI:
10.1039/P19960000953
PDF
Lithium bromide as a new catalyst for carbon–carbon bond formation in the solid state
Dipak Prajapati Kushal C. Lekhok Jagir S. Sandhu and Anil C. Ghosh
pg 959; DOI:
10.1039/P19960000959
PDF
Conference diary

pg viig; DOI:
10.1039/P1996000viig
PDF

Issue 10


Front cover

pg X037; DOI:
10.1039/P199600FX037
PDF
Back cover

pg X039; DOI:
10.1039/P199600BX039
PDF
Contents pages

pg P087; DOI:
10.1039/P199600FP087
PDF
Back matter

pg P095; DOI:
10.1039/P199600BP095
PDF
Chemoenzymatic synthesis of (+)-(4E,15E)-docosa-4,15-dien-1-yn-3-ol, a component of the marine sponge Cribrochalina vasculum
Takehiko Ohtani Keiichi Kikuchi Makoto Kamezawa Hideaki Hamatani Hojun Tachibana Tetsuzo Totani and Yoshinobu Naoshima
pg 961; DOI:
10.1039/P19960000961
PDF
One-pot preparation of isomeric acetyl- and 2,2,2-trifluoroacetyl-azidothiophenes by selective bifunctionalization of dibromothiophenes via halogen–lithio exchange
Piero Spagnolo and Paolo Zanirato
pg 963; DOI:
10.1039/P19960000963
PDF
Two-photon route to N-vinylisoindolinones from isoquinolin-1(2H)-one and electron deficient ethenes
Nader Al-Jalal Michael G. B. Drew and Andrew Gilbert
pg 965; DOI:
10.1039/P19960000965
PDF
Michael addition of N- and O-centred nucleophiles to tethered acrylates. The role of double bond geometry in controlling the diastereoselectivity of cyclisations leading to 2,6-disubstituted tetrahydropyrans and piperidines
Martin G. Banwell Chinh T. Bui Ha T. T. Pham and Gregory W. Simpson
pg 967; DOI:
10.1039/P19960000967
PDF
Solid-phase synthesis of thymosin 10 using a p-cyanotrityl resin. Chemical characterization and immunochemical control of the synthetic peptide
Leondios Leondiadis Irene Vassiliadou Christos Zikos Nikolas Ferderigos Evangelia Livaniou Dionyssis S. Ithakissios and Gregory P. Evangelatos
pg 971; DOI:
10.1039/P19960000971
PDF
Dienophilic thioaldehydes and dithioesters formed by base-catalysed cleavage of alkyl phthalimidosulfanylacetates
Gordon W. Kirby Alistair W. Lochead and Sharon Williamson
pg 977; DOI:
10.1039/P19960000977
PDF
Efficient syntheses of core 1, core 2, and core 3 and core 4 building blocks for SPS of mucin O-glycopeptides based on the N-Dts-method
Ernst Meinjohanns Morten Meldal Axel Schleyer Hans Paulsen and Klaus Bock
pg 985; DOI:
10.1039/P19960000985
PDF
Selective deprotection of phenacyl, benzyl and methyl esters of N-protected amino acids and dipeptides and N-protected amino acids benzyl ester linked to resins with bis(tributyltin) oxide
Claudio J. Salomon Ernesto G. Mata and Oreste A. Mascaretti
pg 995; DOI:
10.1039/P19960000995
PDF
Solid-phase glycopeptide synthesis of tyrosine-glycosylated glycogenin fragments as substrates for glucosylation by glycogenin
Anita M. Jansson Knud J. Jensen Morten Meldal Joseph Lomako Wieslawa M. Lomako Carl Erik Olsen and Klaus Bock
pg 1001; DOI:
10.1039/P19960001001
PDF
Cyclopropanation of tricarbonyl(styrene)chromium(0)and (–)- Ar(1R,2S)-tricarbonyl[2-(trimethylsilyl)styrene] chromium(0)
Susan E. Gibson (née Thomas) Richard Gil Frank Prechtl Andrew J. P. White and David J. Williams
pg 1007; DOI:
10.1039/P19960001007
PDF
Radical initiated reactions of artemisinin derivatives
Bindumadhavan Venugopalan Pravin J. Karnik and Shashikant Shinde
pg 1015; DOI:
10.1039/P19960001015
PDF
Direct and enantiospecific ortho-benzylation of phenols by the Mitsunobu reaction
Shoji Fukumoto Shigeha Fukushi Shinji Terao and Mitsuru Shiraishi
pg 1021; DOI:
10.1039/P19960001021
PDF
Ring-D aromatic phytosteroids; a model for biogenesis by way of carbon radical rearrangement
Stuart P. Green and Donald A. Whiting
pg 1027; DOI:
10.1039/P19960001027
PDF
Pyryliumolates II—generation of and cycloaddition reactions with isoxazole annulated pyryliumolates
Carsten Plüg and Willy Friedrichsen
pg 1035; DOI:
10.1039/P19960001035
PDF
Formation of spiro indane derivatives from hydroxy lactams derived from N-(1-phenylethyl)-phthalimide and -pyridine-2,3-dicarboximide
Abood A. Bahajaj and John M. Vernon
pg 1041; DOI:
10.1039/P19960001041
PDF
The N–N bond as a chiral axis: 3-diacylaminoquinazolinones as chiral acylating agents
Robert S. Atkinson Emma Barker Paul J. Edwards and Gordon A. Thomson
pg 1047; DOI:
10.1039/P19960001047
PDF
Synthesis of (2E,4E)-dienals by double formyl-olefination with an arsonium salt and its application in the syntheses of lipoxygenase metabolites of arachidonic acid
Zhi-Hui Peng Yun-Long Li Wen-Lian Wu Cui-Xian Liu and Yu-Lin Wu
pg 1057; DOI:
10.1039/P19960001057
PDF
Formation of polyheterocyclic systems by reaction of 2-imino-4-methyl-2H-1-benzopyran-3-carbonitrile with active methylene compounds
Conor N. O'Callaghan T. Brain H. McMurry John E. O'Brien Sylvia M. Draper and Deborah J. Wilcock
pg 1067; DOI:
10.1039/P19960001067
PDF
Conference diary

pg ixc; DOI:
10.1039/P19960000ixc
PDF

Issue 11


Front cover

pg X041; DOI:
10.1039/P199600FX041
PDF
Back cover

pg X043; DOI:
10.1039/P199600BX043
PDF
Contents pages

pg P097; DOI:
10.1039/P199600FP097
PDF
Synthesis of novel organic nitrate esters: guanylate cyclase activation and tissue relaxation
Kexin Yang Jennifer D. Artz Jodi Lock Cristina Sanchez Brian M. Bennett Amy B. Fraser and Gregory R. J. Thatcher
pg 1073; DOI:
10.1039/P19960001073
PDF
The first synthesis of Diels–Alder adducts of [60]fullerene with sulfur containing heteroaromatic o-quinodimethanes
Ursula M. Fernández-Paniagua Beatriz M. Illescas Nazario Martín and Carlos Seoane
pg 1077; DOI:
10.1039/P19960001077
PDF
Palladium- and cobalt-mediated cyclisations of halo-polyenes: a comparative study
Amjad Ali G. Bryon Gill Gerald Pattenden Graeme A. Roan and Toh-Seok Kam
pg 1081; DOI:
10.1039/P19960001081
PDF
Polyhalogenated heterocyclic compounds. Part 41. Cycloaddition reactions involving hexafluorobut-2-yne and 1,1,1,2,4,4,4-heptafluorobut-2-ene
Richard D. Chambers Alex J. Roche and Michael H. Rock
pg 1095; DOI:
10.1039/P19960001095
PDF
The design, synthesis and biological evaluation of stable ozonides with antimalarial activity
Luiz-Claudio de Almeida Barbosa David Cutler John Mann M. James Crabbe Geoffrey C. Kirby and David C. Warhurst
pg 1101; DOI:
10.1039/P19960001101
PDF
Asymmetric induction to nitrogen in pyrrolidines and piperidines via radical chemistry
Richard A. Ewin Keith Jones and Christopher G. Newton
pg 1107; DOI:
10.1039/P19960001107
PDF
Stereoselective total synthesis of (–)-pumiliotoxin C by an aqueous intramolecular acylnitroso Diels–Alder approach
Masaichi Naruse Sakae Aoyagi and Chihiro Kibayashi
pg 1113; DOI:
10.1039/P19960001113
PDF
Chiral synthesis of the necic acid components, crobarbatic acid and integerrinecic acid lactone
Toshio Honda Fumihiro Ishikawa and Shin-ichi Yamane
pg 1125; DOI:
10.1039/P19960001125
PDF
Synthesis of (2S,4S)- and (2S,4R)-5,5-dihydroxy[5,5-2H2]leucine by two independent routes
Xavier Durand Piétrick Hudhomme Jeffrey A. Khan and Douglas W. Young
pg 1131; DOI:
10.1039/P19960001131
PDF
Conformational study of the higher [n.n]paracylophanes: evaluation as potential hosts for molecular halogens and benzenes
Mark Mascal Jean-Luc Kerdelhué Andrei S. Batsanov and Michael J. Begley
pg 1141; DOI:
10.1039/P19960001141
PDF
Stereochemistry of the enzymic lactonisation of cis,cis-muconic and 3-methyl-cis,cis-muconic acid
Beining Chen Gordon W. Kirby Ghanakota V. Rao and Ronald B. Cain
pg 1153; DOI:
10.1039/P19960001153
PDF
Reactions of diphenylketene and methylphenylketene with some cis-cyclohexa-3,5-diene-1,2-diol derivatives
Stanley M. Roberts Peter W. Sutton and Lorraine Wright
pg 1157; DOI:
10.1039/P19960001157
PDF
Zinc(II)-catalysed transformation of epoxides to aziridines
Dorte Kühnau Ib Thomsen and Karl Anker Jørgensen
pg 1167; DOI:
10.1039/P19960001167
PDF
Diastereoselectivity in the SE2 reaction of chiral pentadienylsilanes: a test for the relative importance of steric and electronic effects
Ian Fleming Graeme R. Jones Nicholas D. Kindon Yannick Landais Colin P. Leslie Ian T. Morgan Stefan Peukert and Achintya K. Sarkar
pg 1171; DOI:
10.1039/P19960001171
PDF
Stereocontrol of stereogenic centres para on a benzene ring using the SE2 reaction of a pentadienylsilane
Ian Fleming and Colin P. Leslie
pg 1197; DOI:
10.1039/P19960001197
PDF
The 4-azidobenzyloxycarbonyl function; application as a novel protecting group and potential prodrug modification for amines
Roger J. Griffin Elaine Evers Richard Davison Ashleigh E. Gibson Deborah Layton and William J. Irwin
pg 1205; DOI:
10.1039/P19960001205
PDF
Synthesis of inverto-yuehchukene and its 10-(indol-3-yl) isomer. X-Ray structure of (4aRS,10aRS)-1,1,3-trimethyl-1,2,4a,5,10,10a-hexahydroindene [1,2-b]indol-10-one
Kin-Fai Cheng and Man-Ki Cheung
pg 1213; DOI:
10.1039/P19960001213
PDF
Identification of coupling conditions proceeding with low C-terminal epimerization during the assembly of fully protected backbone-substituted peptide segments
Martin Quibell Leonard C. Packman and Tony Johnson
pg 1219; DOI:
10.1039/P19960001219
PDF
Solid-phase assembly of backbone amide-protected peptide segments: an efficient and reliable strategy for the synthesis of small proteins
Martin Quibell Leonard C. Packman and Tony Johnson
pg 1227; DOI:
10.1039/P19960001227
PDF
A new convergent method for porphyrin synthesis based on a 3 + 1 condensation
Arezki Boudif and Michel Momenteau
pg 1235; DOI:
10.1039/P19960001235
PDF
Synthesis and stereostructure–activity relationship of a synthetic pyrethroid, 2-chloro-1-methyl-3-phenylcyclopropylmethyl-3-phenoxybenzyl ether
Yoshinori Nishii Ken-ichi Wakimura Toru Tsuchiya Shogo Nakamura and Yoo Tanabe
pg 1243; DOI:
10.1039/P19960001243
PDF
Reaction of metallo-2-nitro-5,10,15,20-tetraphenylporphyrins with oxyanions. Temperature-dependent competition between nucleophilic addition and single-electron transfer processes
Maxwell J. Crossley and Lionel G. King
pg 1251; DOI:
10.1039/P19960001251
PDF
Novel indole-ring formation by thermolysis of 2-(N-acylamino)-benzylphosphonium salts. Effective synthesis of 2-trifluoromethylindoles
Kazuyuki Miyashita Katsunori Kondoh Katsutoshi Tsuchiya Hideto Miyabe and Takeshi Imanishi
pg 1261; DOI:
10.1039/P19960001261
PDF
Synthesis of 15,15-dialkylestradiols
James R. Bull and Michiel C. Loedolff
pg 1269; DOI:
10.1039/P19960001269
PDF
Syntheses and chemical and physical properties of thiophenetriptycenes
Akihiko Ishii Kiyoto Maeda Maki Kodachi Noriko Aoyagi Keiko Kato Teruo Maruta Masamatsu Hoshino and Juzo Nakayama
pg 1277; DOI:
10.1039/P19960001277
PDF
An approach to modified heterocyclic analogues of huperzine A and isohuperzine A. Synthesis of the pyrimidone and pyrazole analogues, and their anticholinesterase activity
Alan P. Kozikowski Giuseppe Campiani Vito Nacci Alessandro Sega Ashima Saxena and Bhupendra P. Doctor
pg 1287; DOI:
10.1039/P19960001287
PDF
Self-addition products from the alkylation of amino acid-derived oxazolidinones: X-ray molecular structures of (2R,4S,1S)-3-benzoyl-4-[benzoylamino(phenyl)methyl]-4-benzyl-2-phenyl-1,3-oxazolidin-5-one, (2R,4S,1S)- and (2R,4S,1R)-3-benzoyl-4-[benzoylamino(phenyl)methyl]-4-isopropyl-2-phenyl-1,3-oxazolidin-5-one
Andrew D. Abell Jane M. Taylor and Mark D. Oldham
pg 1299; DOI:
10.1039/P19960001299
PDF
Synthesis of chiral bicyclo[2.2.2]oct-5-en-2-ones via an intramolecular alkylation reaction
Adusumilli Srikrishna G. Veera Raghava Sharma Savariappan Danieldoss and Parthasarathy Hemamalini
pg 1305; DOI:
10.1039/P19960001305
PDF
Corrigenda
Vijay Nair Jessy Mathew Tomohiro Okawa Shoji Eguchi and Akikazu Kakehi
pg 1313; DOI:
10.1039/P19960001313
PDF
Conference diary

pg ixd; DOI:
10.1039/P19960000ixd
PDF

Issue 12


Front cover

pg X045; DOI:
10.1039/P199600FX045
PDF
Back cover

pg X047; DOI:
10.1039/P199600BX047
PDF
Contents pages

pg P105; DOI:
10.1039/P199600FP105
PDF
Back matter

pg P113; DOI:
10.1039/P199600BP113
PDF
Total synthesis of the virginiamycin antibiotic 14,15-anhydropristinamycin IIB
David A. Entwistle Stuart I. Jordan John Montgomery and Gerald Pattenden
pg 1315; DOI:
10.1039/P19960001315
PDF
An alternative isoxazole route to -alkoxycarbonyl--diketones
Raymond C. F. Jones Stephen H. Dunn and Kathryn A. M. Duller
pg 1319; DOI:
10.1039/P19960001319
PDF
Short synthesis of the furanofuran sub-unit of the toxin erythroskyrine
Raffaella Rossin Peter R. Jones Patrick J. Murphy and W. Roger Worsley
pg 1323; DOI:
10.1039/P19960001323
PDF
New anthracycline disaccharides. Synthesis of L-daunosaminyl-(1 4)-2-deoxy-L-rhamnosyl and of L-daunosaminyl-(1 4)-2-deoxy-L-fucosyl daunorubicin analogues
Fabio Animati Federico Arcamone Marco Berettoni Amalia Cipollone Maurizio Franciotti and Paolo Lombardi
pg 1327; DOI:
10.1039/P19960001327
PDF
Synthesis of novel piperideine- and pyridine-containing long-chain fatty ester derivatives from methyl iso-ricinoleate
Marcel S. F. Lie Ken Jie and Mohammed Khysar Pasha
pg 1331; DOI:
10.1039/P19960001331
PDF
N-formimidoyl analogues of distamycin
Giovanna Di Pietro Giuseppe Giannini Elisabetta M. Iafrate Edith Monteagudo Mariella Dentini Fabio Animati Paolo Lombardi and Federico Arcamone
pg 1333; DOI:
10.1039/P19960001333
PDF
Stereoselective rearrangement of 5,6-epoxy carotenoid model compounds
Yumiko Yamano Chisato Tode and Masayoshi Ito
pg 1337; DOI:
10.1039/P19960001337
PDF
Azoles. Part 13. Synthesis and bromine lithium exchange reactions of some 1-substituted 4,5-dibromo-1H-1,2,3-triazoles and 2-substituted 4,5-dibromo-2H-1,2,3-triazoles
Brian Iddon and Martin Nicholas
pg 1341; DOI:
10.1039/P19960001341
PDF
Reactions of acyl isothiocyanates with 9-diazofluorene: a route to macromolecules having pairs of orthogonal fluorene groups
Gerrit L'abbé Agna Francis and Wim Dehaen
pg 1349; DOI:
10.1039/P19960001349
PDF
Asymmetric syntheses of isostegane derivatives using trivalent iodine reagents
Andrew Pelter Robert S. Ward and Atef Abd-el-Ghani
pg 1353; DOI:
10.1039/P19960001353
PDF
v-Triazolines. Part 37. Rearrangement reactions of 5-amino-1-(2-formyl-, -benzoyl-, -cyano-aryl)--triazolines: new synthesis of 2-amino- and 2,4-diamino-quinolines and 2,4-diamino-1,7-naphthyridines
Egle M. Beccalli Emanuela Erba Maria Luisa Gelmi and Donato Pocar
pg 1359; DOI:
10.1039/P19960001359
PDF
Synthesis of D-2-deoxy-myo-inositol 1,3,4,5-tetrakisphosphate from D-glucose
David J. Jenkins Didier Dubreuil and Barry V. L. Potter
pg 1365; DOI:
10.1039/P19960001365
PDF
Ketone-directed peracid epoxidation of cyclic alkenes
Alan Armstrong Paul A. Barsanti Paul A. Clarke and Anthony Wood
pg 1373; DOI:
10.1039/P19960001373
PDF
Simple reduction of ferrocenyl aldehydes and ketones by sodium boranuide in trifluoroacetic acid: new, efficient, general preparation of alkylferrocenes
Sukanta Bhattacharyya
pg 1381; DOI:
10.1039/P19960001381
PDF
The total synthesis of the diepoxycyclohexanone antibiotic aranorosin and novel synthetic analogues
Alexander McKillop Lee McLaren Richard J. K. Taylor Robert J. Watson and Norman J. Lewis
pg 1385; DOI:
10.1039/P19960001385
PDF
The synthesis of precisely structured polyurethanes. Part 2. Chain building methodology
Maurice H. George Helen C. Hailes and David A. Widdowson
pg 1395; DOI:
10.1039/P19960001395
PDF
A new facet of the reaction of nitro heteroaromatic compounds with ethyl isocyanoacetate
Takashi Murashima Ken-ichi Fujita Kazuo Ono Takuji Ogawa Hidemitsu Uno and Noboru Ono
pg 1403; DOI:
10.1039/P19960001403
PDF
Addition of organolithium reagents to -(trifluoromethyl)styrene: concise synthesis of functionalised gem-difluoroalkenes
Jean-Pierre Bégué Danièle Bonnet-Delpon and Michael H. Rock
pg 1409; DOI:
10.1039/P19960001409
PDF
Enhancement of tyrosinase activity by macrocycles in the oxidation of p-cresol in organic solvents
Jaap Broos Renate Arends Gerrit B. van Dijk Willem Verboom Johan F. J. Engbersen and David N. Reinhoudt
pg 1415; DOI:
10.1039/P19960001415
PDF
Metabolites of the higher fungi. Part 29. Maldoxin, maldoxone, dihydromaldoxin, isodihydromaldoxin and dechlorodihydromaldoxin. A spirocyclohexadienone, a depsidone and three diphenyl ethers: keys in the depsidone biosynthetic pathway from a member of the fungus genus Xylaria
Monilola O. Adeboya Raymond L. Edwards Thomas Lassøe Derek J. Maitland Len Shields and Anthony J. S. Whalley
pg 1419; DOI:
10.1039/P19960001419
PDF
Synthesis of derivatives of (2S,4S)-4-hydroxy-2,5-dimethyl-3-oxohexanoic acid, a constituent of the didemnins
Isabel González Gemma Jou Josep Maria Caba Fernando Albericio Paul Lloyd-Williams and Ernest Giralt
pg 1427; DOI:
10.1039/P19960001427
PDF
Electrochemical synthesis of chroman and euglobal skeletons via cycloaddition reaction of o-quinone methides and alkenes
Kazuhiro Chiba Junko Sonoyama and Masahiro Tada
pg 1435; DOI:
10.1039/P19960001435
PDF
Studies in the cycloproparene series: oxygen-containing 1H-cyclopropa[b]naphthalenes and their methylidene derivatives
Brian Halton Andrew J. Kay Zha Zhi-Mei Roland Boeseb and Thomas Haumann
pg 1445; DOI:
10.1039/P19960001445
PDF
Metal-assisted reactions. Part 25. Heterogeneous and homogeneous catalytic transfer hydrogenolysis of allyloxytetrazoles to yield alkenes or alkanes
M. Lurdes S. Cristiano Robert A. W. Johnstone and Peter J. Price
pg 1453; DOI:
10.1039/P19960001453
PDF
Photoreaction of homobenzoquinones with amine donors
Hiroshi Moriwaki Takashi Matsumoto Toshikazu Nagai and Takumi Oshima
pg 1461; DOI:
10.1039/P19960001461
PDF
Phosphane ligands with two binding sites of differing hardness for enantioselective Grignard cross coupling
Andreas Terfort and Henri Brunner
pg 1467; DOI:
10.1039/P19960001467
PDF
Synthesis of 4-phosphazenyl-2,3-dihydropyrrol-2-ones and 5-phosphazenyl-2-pyridones from -[(N-acyl)phosphazenyl]enamines and dimethyl acetylenedicarboxylate
Elvira Pelàez-Arango and Fernando López-Ortiz
pg 1481; DOI:
10.1039/P19960001481
PDF
Oxidative addition of 1,3-dicarbonyl compounds to alkenes mediated by cerium(IV) ammonium nitrate and manganese(III) acetate: a comparative study
Vijay Nair Jessy Mathew and K. V. Radhakrishnan
pg 1487; DOI:
10.1039/P19960001487
PDF
Conference diary

pg ixe; DOI:
10.1039/P19960000ixe
PDF

Issue 13


Front cover

pg X049; DOI:
10.1039/P199600FX049
PDF
Journals bulletin

pg X051; DOI:
10.1039/P1996000X051
PDF
Back cover

pg X055; DOI:
10.1039/P199600BX055
PDF
Contents pages

pg P115; DOI:
10.1039/P199600FP115
PDF
Back matter

pg P121; DOI:
10.1039/P199600BP121
PDF
Radical-chain reactions of sulfonyl azides and of ethyl azidoformate with allylstannanes: homolytic allylation at nitrogen
Hai-Shan Dang and Brian P. Roberts
pg 1493; DOI:
10.1039/P19960001493
PDF
Reaction of 4-picoline(2,2 :6,2-terpyridine)platinum(II) with nucleosides
Gordon Lowe and Tirayut Vilaivan
pg 1499; DOI:
10.1039/P19960001499
PDF
On the stereoselection of iodolactonizations of 3-silyloxyalk-5-enoic acids
Simon B. Bedford Garry Fenton David W. Knight and Duncan E. Shaw
pg 1505; DOI:
10.1039/P19960001505
PDF
A new silicon-mediated elimination–rearrangement
Stefano Menichetti and Charles J. M. Stirling
pg 1511; DOI:
10.1039/P19960001511
PDF
Chemistry of insect antifeedants from Azadirachta indica(part 20): synthesis of biologically active, simple analogues of azadirachtin, containing the hydroxytetrahydrofurancarboxylate hemiketal moiety
María L. de la Puente Robert B. Grossman Steven V. Ley Monique S. J. Simmonds and Wally M. Blaney
pg 1517; DOI:
10.1039/P19960001517
PDF
Chemistry of insect antifeedants from Azadirachta indica(part 21): synthesis of model compounds of azadirachtin using a decalin framework as a functional group scaffolding
María L. de la Puente Steven V. Ley Monique S. J. Simmonds and Wally M. Blaney
pg 1523; DOI:
10.1039/P19960001523
PDF
On the stereochemical outcome of the reaction between (–)-chorismic acid and diazomethane: absolute proof of stereochemistry of the major pyrazoline by X-ray crystallography of a cyclopropane based derivative
Harry Adams Neil A. Bailey Martyn Frederickson Edwin Haslam Gareth M. Davies and David A. Jude
pg 1531; DOI:
10.1039/P19960001531
PDF
Towards the total synthesis of cyclo[n]carbons and the generation of cyclo[6]carbon
George A. Adamson and Charles W. Rees
pg 1535; DOI:
10.1039/P19960001535
PDF
One-pot synthesis of tetrasubstituted pyrazoles—proof of regiochemistry
Ulf Hanefeld Charles W. Rees Andrew J. P. White and David J. Williams
pg 1545; DOI:
10.1039/P19960001545
PDF
New linked macrocyclic systems derived from selectively protected S2N2 macrocycles
Andrew M. Groth Leonard F. Lindoy and George V. Meehan
pg 1553; DOI:
10.1039/P19960001553
PDF
Parasite glycoconjugates. Part 5. Blockwise approach to oligo(glycosyl phosphates): chemical synthesis of a terminal tris(glycobiosyl phosphate) fragment of Leishmania donovani antigenic lipophosphoglycan
Andrei V. Nikolaev Trevor J. Rutherford Michael A. J. Ferguson and John S. Brimacombe
pg 1559; DOI:
10.1039/P19960001559
PDF
Tandem Beckmann and Huisgen–White rearrangement as an alternative to the Baeyer–Villiger oxidation of the bicyclo[3.3.1]nonane system: first asymmetric synthesis of (–)-dihydropalustramic acid. X-Ray molecular structure of 2-ethyl-9-phenylsulfonyl-9-azabicyclo[3.3.1]nonan-3-one
Osamu Muraoka Bao-Zhong Zheng Kazuhito Okumura Genzoh Tanabe Takefumi Momose and Conrad Hans Eugster
pg 1567; DOI:
10.1039/P19960001567
PDF
New insight into the pyruvate decarboxylase-catalysed formation of lactaldehyde from H–D exchange experiments: a water proof active site
Mario Lobell and David H. G. Crout
pg 1577; DOI:
10.1039/P19960001577
PDF
Synthesis and evaluation of photolabile sulfonamides as potential reagents for rapid photorelease of neuroactive amines
John E. T. Corrie and George Papageorgiou
pg 1583; DOI:
10.1039/P19960001583
PDF
A study of solvent effect on photochemically induced reations between pyridinedicarbonitriles and alkenes: an easy approach to the synthesis of cyclopenta [b or c]pyridines
Rosanna Bernardi Tullio Caronna Daniela dal Pio Luogo Sergio Morrocchi Gabriella Poggi and Bruno M. Vittimberga
pg 1593; DOI:
10.1039/P19960001593
PDF
Syntheses of some -substituted alkyne porphyrins related to protoporphyrin-IX
Xuqin Jiang and Kevin M. Smith
pg 1601; DOI:
10.1039/P19960001601
PDF
Nucleoside adducts of vinylporphyrins and vinylchlorins
Xuqin Jiang Ravindra K. Pandey and Kevin M. Smith
pg 1607; DOI:
10.1039/P19960001607
PDF
1,2,3-Trizolium-1-unsubstituted methanides, carbon analogues of triazole-N-oxides: a 1,3-dipole cascade from 1,2,3-triazolium-1-methanide to 1,2,4-triazinium-4-methanide: new routes to pyrrolo[1,2-c][1,2,3]triazoles, pyrrolo[1,2-d][1,2,4]triazines and substituted 1-aminopyrroles. Azolium 1,3-dipoles
Richard N. Butler Peter D. McDonald Patrick McArdle and Desmond Cunningham
pg 1617; DOI:
10.1039/P19960001617
PDF
Tricyclic phenanthrene systems: substituted phenanthro[9,10-e]-1,2,3-triazines and fused phenanthro-azolo-1,2,3-triazoles from cycloaddition—rearrangement sequences of 9,10-bisarylazophenanthrenes with 2-dipolarophiles. Azolium 1,3-dipoles
Richard N. Butler Fiona A. Lysaght Peter D. McDonald Carmel S. Pyne Patrick McArdle and Desmond Cunningham
pg 1623; DOI:
10.1039/P19960001623
PDF
Novel reactions of N-sulfonylamines with 3-dimethylamino-2H-azirines. Competitive formation of 1,2,5-thiadiazoles, 1,2,3-oxathiazoles and acrylamidines. X-Ray molecular structure of N-(4-dimethylamino-5-methyl-2-oxo-5-phenyl-5H-1,26,3-oxathiazol-2-ylidene)benzamide
Ingo Tornus Ernst Schaumann and Gunadi Adiwidjaja
pg 1629; DOI:
10.1039/P19960001629
PDF
A versatile process for the syntheses of very long chain alkanes, functionalised derivatives and some branched chain hydrocarbons
Gerald M. Brooke Simon Burnett Shahid Mohammed David Proctor and Mark C. Whiting
pg 1635; DOI:
10.1039/P19960001635
PDF
Conference diary

pg viih; DOI:
10.1039/P1996000viih
PDF

Issue 14


Front cover

pg X057; DOI:
10.1039/P199600FX057
PDF
Back cover

pg X059; DOI:
10.1039/P199600BX059
PDF
Contents pages

pg P123; DOI:
10.1039/P199600FP123
PDF
Back matter

pg P131; DOI:
10.1039/P199600BP131
PDF
A versatile synthesis of benzo[c]phenanthridine alkaloids
Graham R. Geen Inderjit S. Mann M. Valerie Mullane and Alexander McKillop
pg 1647; DOI:
10.1039/P19960001647
PDF
Novel approach to the synthesis of the aromatase inhibitor 4-hydroxyandrost-4-ene-3,17-dione (4-OHA)
Elisiario J. Tavares da Silva Maria L. Sá e Melo and André S. Campos Neves
pg 1649; DOI:
10.1039/P19960001649
PDF
(Nonracemic) thiols and ZnII. Structural and catalytic aspects of some natural and non-natural zinc thiolates
Richard M. Kellogg and Robert P. Hof
pg 1651; DOI:
10.1039/P19960001651
PDF
Elemental fluorine. Part 4. Use of elemental fluorine for the halogenation of aromatics
Richard D. Chambers Christopher J. Skinner Malcolm J. Atherton and John S. Moilliet
pg 1659; DOI:
10.1039/P19960001659
PDF
Synthesis and configurational assignments of 3-substituted 2-deoxy-4-thio-D-erythro-pentafuranose derivatives
Houssine Ait-Sir Nour-Eddine Fahmi Gérard Goethals Gino Ronco Bougrine Tber Pierre Villa David F. Ewing and Grahame Mackenzie
pg 1665; DOI:
10.1039/P19960001665
PDF
Stereoselective addition of organometallic reagents to N-(tosyl)vinylsulfoximines
Richard F. W. Jackson Andrew D. Briggs Paul A. Brown William Clegg Mark R. J. Elsegood and Christopher Frampton
pg 1673; DOI:
10.1039/P19960001673
PDF
Membrane-permeant analogues of the putative second messenger myo-inositol 3,4,5,6-tetrakisphosphate
Stefan Roemer Christoph Stadler Marco T. Rudolf Bernd Jastorff and Carsten Schultz
pg 1683; DOI:
10.1039/P19960001683
PDF
Conversion of xanthyrones into glutaconic anhydride–pyrone (GP) compounds in strong acid media: selective deuteriation as between chelated and unchelated acetyls
Leslie Crombie and Roderick V. Dove
pg 1695; DOI:
10.1039/P19960001695
PDF
Polyaza heterocycles. Part 3. Halogenation of 1-substituted quinoxalino[2,3-c]cinnolines: mechanistic implications
Ian W. Harvey David M. Smith and Charles R. White
pg 1699; DOI:
10.1039/P19960001699
PDF
Reaction of ynolate anions derived from silylketenes with electrophiles: a facile preparation of silyl ynol ethers and functionalized silylketenes
Shuji Akai Shinji Kitagaki Tadaatsu Naka Kiyoshi Yamamoto Yasunori Tsuzuki Keita Matsumoto and Yasuyuki Kita
pg 1705; DOI:
10.1039/P19960001705
PDF
Selective ipso-nitration of tert-butylcalix[4]arene 1,3-diethers: X-ray structure of an unexpected side product
Oliver Mogck Volker Böhmer George Ferguson and Walter Vogt
pg 1711; DOI:
10.1039/P19960001711
PDF
Synthesis of L-scyllo-inositol 1,2,4-trisphosphate, scyllo-inositol 1,2,4,5-tetrakisphosphate and phosphorothioate and DL-2-deoxy-2-fluoro-myo-inositol 1,4,5-trisphosphate: optical resolution of DL-1-O-allyl-3,6-di-O-benzyl-4,5-O-isopropylidene-scyllo-inositol
Dethard Lampe Changsheng Liu Mary F. Mahon and Barry V. L. Potter
pg 1717; DOI:
10.1039/P19960001717
PDF
Studies on the sharpless asymmetric epoxidation of unsymmetrical divinylmethanols
Toshio Honda Hirotake Mizutani and Kazuo Kanai
pg 1729; DOI:
10.1039/P19960001729
PDF
Novel and practical preparation of -fluoro-functionalized esters from fluoroiodoacetates
Chengxin Zhi and Qing-Yun Chen
pg 1741; DOI:
10.1039/P19960001741
PDF
Studies on Rubia akane(RA) derivatives. Part 10. Backbone transformation of RA-VII, an antitumour cyclic hexapeptide, through thionation. X-Ray crystal structure of [Tyr-3-(CH2NH)-Ala-4]RA-VII
Yukio Hitotsuyanagi Yuji Matsumoto Shin-ichi Sasaki Jin Suzuki Koichi Takeya Kentaro Yamaguchi and Hideji Itokawa
pg 1749; DOI:
10.1039/P19960001749
PDF
Chemical and enzyme-catalysed syntheses of enantiopure epoxide and diol derivatives of chromene, 2,2-dimethylchromene, and 7-methoxy-2,2-dimethylchromene (precocene-1)
Derek R. Boyd Narain D. Sharma Rosemary Boyle Timothy A. Evans John F. Malone Kenneth M. McCombe Howard Dalton and Jagdeep Chima
pg 1757; DOI:
10.1039/P19960001757
PDF
New Diels–Alder reactions of 3-vinylindoles with an aryne: selective access to functionalized [a]anellated carbazoles
Eugenia Gonzalez Ulf Pindur and Dieter Schollmeyer
pg 1767; DOI:
10.1039/P19960001767
PDF
Conference diary

pg ixf; DOI:
10.1039/P19960000ixf
PDF

Issue 15


Front cover

pg X061; DOI:
10.1039/P199600FX061
PDF
Back cover

pg X063; DOI:
10.1039/P199600BX063
PDF
Contents pages

pg P135; DOI:
10.1039/P199600FP135
PDF
Brasiliquinones A–C, new cytotoxic benz[a]anthraquinones with an ethyl group at C-3 from actinomycete Nocardia brasiliensis
Masashi Tsuda Hiroyasu Sato Yasushi Tanaka Katsukiyo Yazawa Yuzuru Mikami Takuma Sasaki and Jun'ichi Kobayashi
pg 1773; DOI:
10.1039/P19960001773
PDF
DMSO–Ac2O promoted nitration of isoquinolines. One-step synthesis of 1-nitroisoquinolines under mild conditions
Woonphil Baik Sangmin Yun Jong Uk Rhee and Glen A. Russell
pg 1777; DOI:
10.1039/P19960001777
PDF
Preparation and reactions of 2-pyridyltellurium derivatives
Yoshinori Kondo Manabu Shilai Masanobu Uchiyama and Takao Sakamoto
pg 1781; DOI:
10.1039/P19960001781
PDF
Synthesis, electrochemical and chemical oxidations, and peri selenium participation of macrocyclic polyselenides containing naphthalene rings
Hisashi Fujihara Masayoshi Yabe and Naomichi Furukawa
pg 1783; DOI:
10.1039/P19960001783
PDF
Anti-tumour heterocycles. Part xiv. A new route to pyrrolo-[3,2-f]indoles and the novel pyrrolo[3,2-f; 4,5-f]diindole system
Laddawan Chunchatprasert and Patrick V. R. Shannon
pg 1787; DOI:
10.1039/P19960001787
PDF
A synthesis of 18-O-methyl mycalamide B
Philip Kocienski Piotr Raubo Justin K. Davis F. Thomas Boyle Donna E. Davies and Audrey Richter
pg 1797; DOI:
10.1039/P19960001797
PDF
Diels–Alder reactions of N-sulfonyl substituted aza-ortho-xylylenes generated from the corresponding 1,4-dihydro-2H-3,1-benzoxazin-2-one derivatives
Roberto Consonni Piero Dalla Croce Raffaella Ferraccioli and Concetta La Rosa
pg 1809; DOI:
10.1039/P19960001809
PDF
Aluminium chloride2-isocyanatobenzoyl chloride complex: crystal structure and reactivity
Franca Bigi Giovanni Sartori Raimondo Maggi Claudia Valerio-Papa Elena Marzi Maurizio Lanfranchi and Maria Angela Pellinghelli
pg 1815; DOI:
10.1039/P19960001815
PDF
Synthesis of bridged azabicyclic compounds using radical translocation reactions of 1-(o-halogenobenzoyl)-2-(prop-2-enyl)- and -(prop-2-ynyl)-piperidines
Masazumi Ikeda Yasuhiro Kugo and Tatsunori Sato
pg 1819; DOI:
10.1039/P19960001819
PDF
Metal-assisted fragmentation of N-aryl- and -alkyl-N-trimethyl-silylaminosulfur chlorides and N-aryl- and -alkyl-aminosulfur chlorides in the presence of conjugated dienes: synthesis and reactivity of 2-substituted-3,6-dihydro-1,2-thiazines
Martin R. Bryce Antony Chesney Graham N. McKelvey Andrei S. Batsanov Judith A. K. Howard and Martin Anderson
pg 1825; DOI:
10.1039/P19960001825
PDF
Oxidation of didehydro--amino acids as a route to -hydroxy-or -amino-pyruvic derivatives and to -acylglycinates
Benoît Miossec Hélène Rudyk Loïc Toupet Renée Danion-Bougot and Daniel Danion
pg 1833; DOI:
10.1039/P19960001833
PDF
Novel construction of 5-methylenepyrrol-2-ones by intramolecular cyclization of selenium-stabilized alkynyl amides
Mitsuhiro Yoshimatsu Keigo Machida Takayo Fuseya Hiroshi Shimizu and Tadashi Kataoka
pg 1839; DOI:
10.1039/P19960001839
PDF
Synthesis of 3,4,5,6-tetrakisphosphates of DL-1,2-dideoxy-1,2-difluoro-myo-inositol and DL-1,2-dideoxy-1,2-difluoro-scyllo-inositol as analogues of DL-myo-inositol 3,4,5,6-tetrakisphosphate
Kevin R. H. Solomons Sally Freeman David R. Poyner and Farid Yafai
pg 1845; DOI:
10.1039/P19960001845
PDF
Synthesis of 3-(2,2,2-trifluoroethylidene)-lactams. First examples of 1,3-dipolar cycloaddition with diazomethane and N-methyl--phenylnitrone
Jean-Philippe Bouillon Zdenek Janousek Heinz G. Viehe Bernard Tinant and Jean-Paul Declercq
pg 1853; DOI:
10.1039/P19960001853
PDF
Ritter reactions. Part 11. The diverse reactivity of 5,10-(azenometheno)-5H-dibenzo[a,d]cyclohepten-11-yl amides with dimethyl acetylenedicarboxylate
Djamal Djaidi Roger Bishop Donald C. Craig and Marcia L. Scudder
pg 1859; DOI:
10.1039/P19960001859
PDF
Comparison of microbiologically and enzymatically mediated Baeyer–Villiger oxidations: synthesis of optically active caprolactones
Véronique Alphand Roland Furstoss Sandrine Pedragosa-Moreau Stanley M. Roberts and Andrew J. Willetts
pg 1867; DOI:
10.1039/P19960001867
PDF
Cathodic carbonylation. Synthesis of aliphatic aldehydes using an electroreductively generated iron-carbonyl anion
Kunihisa Yoshida and Hideki Kuwata
pg 1873; DOI:
10.1039/P19960001873
PDF
Enantioselective preparation of 1,3-dithiane 1-oxides by asymmetric oxidation of 1,3-dithianes bearing a chiral auxiliary
Yoshihiko Watanabe Yojiro Ono Shigefumi Hayashi Yoshio Ueno and Takeshi Toru
pg 1879; DOI:
10.1039/P19960001879
PDF
Intramolecular O–H hydrogen bond found in [2.2]metacyclophane systems: spectral properties and X-ray crystallographic analysis of 8-hydroxymethyl[2.2]metacyclophanes
Tsutomu Ishi-i Tsuyoshi Sawada Shuntaro Mataka and Masashi Tashiro
pg 1887; DOI:
10.1039/P19960001887
PDF
Studies on organophosphorus compounds. Part 96. Nucleophilicity of the isocyano carbon atom in diethyl isocyanomethylphosphonate. First generation of a phosphorylated nitrile ylide and new syntheses of pyrrolinephosphonates and pyrrolephosphonates
Wei-Sheng Huang Yi-Xin Zhang and Chengye Yuan
pg 1893; DOI:
10.1039/P19960001893
PDF
Uncatalysed (thermal) and Lewis acid-promoted asymmetric hetero-Diels–Alder reaction of 1-thiabuta-1,3-dienes (thiochalcones) with di-(–)-menthyl fumarate. Configuration determination by X-ray crystallographic analysis of (2S,3R,4R)-(+)-2,3-bis[(–)-menthoxycarbonyl]-4,6-diphenyl-3,4-dihydro-2H-thiopyran and conversion of cycloadducts into optically pure diols
Takao Saito Hironari Fujii Satoshi Hayashibe Teruki Matsushita Hideo Kato and Kimiko Kobayashi
pg 1897; DOI:
10.1039/P19960001897
PDF
A new synthesis of 1-phenylthio- and 1-alkylamino-4-nitrobuta-1,3-dienes
Noboru Ono Koji Matsumoto Takuji Ogawa Hiroyuki Tani and Hidemitsu Uno
pg 1905; DOI:
10.1039/P19960001905
PDF
Conference diary

pg ixg; DOI:
10.1039/P19960000ixg
PDF

Issue 16


Front cover

pg X065; DOI:
10.1039/P199600FX065
PDF
Back cover

pg X067; DOI:
10.1039/P199600BX067
PDF
Contents pages

pg P143; DOI:
10.1039/P199600FP143
PDF
Back matter

pg P151; DOI:
10.1039/P199600BP151
PDF
A convenient one-pot synthesis of cystine-containing peptides from protected peptidyl resins using the trimethylsilyl chloride–dimethyl sulfoxide–trifluoroacetic acid system
Hirokazu Tamamura Tsunehito Ishihara Akira Otaka Takaki Koide Kengo Miyoshi Toshiro Ibuka and Nobutaka Fujii
pg 1911; DOI:
10.1039/P19960001911
PDF
Preparation and palladium-catalysed cross-coupling reactions of 3- and 4-tributylstannylfuran-2(5H)-ones
Gregory J. Hollingworth Gemma Perkins and Joseph Sweeney
pg 1913; DOI:
10.1039/P19960001913
PDF
Glycosidase-catalysed oligosaccharide synthesis of di-, tri- and tetra-saccharides using the N-acetylhexosaminidase from Aspergillus oryzae and the -galactosidase from Bacillus circulans
Suddham Singh Michaela Scigelova Gabin Vic and David H. G. Crout
pg 1921; DOI:
10.1039/P19960001921
PDF
Preparation and palladium-catalysed arylation of indolylzinc halides
Takao Sakamoto Yoshinori Kondo Nobuo Takazawa and Hiroshi Yamanaka
pg 1927; DOI:
10.1039/P19960001927
PDF
Kinetic resolution in asymmetric anti aldol reactions of branched and straight chain racemic 2-phenylsulfanyl aldehydes: asymmetric synthesis of cyclic ethers and lactones by phenylsulfanyl migration
Kelly Chibale and Stuart Warren
pg 1935; DOI:
10.1039/P19960001935
PDF
Elemental fluorine. Part 5. Reactions of 1,3-dithiolanes and thioglycosides with fluorine–iodine mixtures
Richard D. Chambers Graham Sandford Matthew E. Sparrowhawk and Malcolm J. Atherton
pg 1941; DOI:
10.1039/P19960001941
PDF
Synthesis and optical resolution of naphthalene-containing inherently chiral calix[4]arenes derived by intramolecular ring closure or stapling of proximal phenyl units
Atsushi Ikeda Makoto Yoshimura Pavel Lhotak and Seiji Shinkai
pg 1945; DOI:
10.1039/P19960001945
PDF
Aziridination of ,-unsaturated esters bearing allylic hydroxy groups with 3-acetoxyaminoquinazolinones: evidence for a mechanism comprising Michael addition–SN2 nucleophilic displacement of acetoxy for aziridination of ,-unsaturated esters
Robert S. Atkinson and Paul J. Williams
pg 1951; DOI:
10.1039/P19960001951
PDF
Reactivity of conjugated azoalkenes towards -amino acid ethyl esters
Silvano Bozzini Fulvia Felluga Giorgio Nardin Alessandro Pizzioli Giuliana Pitacco and Ennio Valentin
pg 1961; DOI:
10.1039/P19960001961
PDF
First synthesis, X-ray structure analysis and reactions of alkenyltriphenylbismuthonium salts
Yoshihiro Matano Masanori Yoshimune Nagao Azuma and Hitomi Suzuki
pg 1971; DOI:
10.1039/P19960001971
PDF
Sesquiterpene lactones from feverfew, Tanacetum parthenium: isolation, structural revision, activity against human blood platelet function and implications for migraine therapy
Martin J. Hewlett (the late) Michael J. Begley W. Antoinette Groenewegen Stan Heptinstall David W. Knight Jane May Umit Salan and Dane Toplis
pg 1979; DOI:
10.1039/P19960001979
PDF
Oxidative rearrangement of 2-hydroxychalcones having no substituent at the 3- and 5-positions with thallium(III) nitrate in methanol
Tokunaru Horie Yasuhiko Kawamura Chikako Sakai Ayako Akita Masahiro Sasagawa and Toshihide Yamada
pg 1987; DOI:
10.1039/P19960001987
PDF
Selective reduction of mixed anhydrides of carboxylic acids to alcohols using borohydride exchange resin (BER)–nickel acetate
B. P. Bandgar R. K. Modhave P. P. Wadgaonkar and A. R. Sande
pg 1993; DOI:
10.1039/P19960001993
PDF
Synthesis of novel tetrathiafulvalene derivatives with thiacrowns
Michael Wagner Dennis Madsen Jan Markussen Sine Larsen Kjeld Schaumburg Karl-Heinz Lubert Jan Becher and Ruth-Maria Olk
pg 1995; DOI:
10.1039/P19960001995
PDF
Studies on pyrimidine-annelated heterocycles: synthesis of novel pyrazolo[3,4:4,5]pyrido[2,3-d]pyrimidines by intramolecular 1,3-dipolar cycloadditions
Bipul Baruah Dipak Prajapati Jagir S. Sandhu and Anil C. Ghosh
pg 1999; DOI:
10.1039/P19960001999
PDF
Synthesis of benzocycloheptenones by 1,3-dipolar additions of 2-(1,3-benzodioxol-5-ylmethyl)-4-hydroxy-3-methoxy-carbonylisoquinolin-2-ium chloride with dipolarophiles
Jeremy J. Edmunds Xue-Min Cheng and Brian Tobias
pg 2005; DOI:
10.1039/P19960002005
PDF
Characterisation of stress protein LysU. Enzymic synthesis of diadenosine 5,5-P1,P4-tetraphosphate (Ap4A) analogues by LysU
Maria-Elena Theoclitou E. Pernilla L. Wittung Alison D. Hindley Talal S. H. El-Thaher and Andrew D. Miller
pg 2009; DOI:
10.1039/P19960002009
PDF
Isolation and structural elucidation of the 11-residue peptaibol antibiotic, harzianin HK VI
Sylvie Rebuffat Sanae Hlimi Yann Prigent Christophe Goulard and Bernard Bodo
pg 2021; DOI:
10.1039/P19960002021
PDF
Synthesis of esters of the potent anti-bacterial trinems and analogues
P. Mark Jackson Stanley M. Roberts Silvia Davalli Daniele Donati Carla Marchioro Alcide Perboni Stefano Proviera and Tino Rossi
pg 2029; DOI:
10.1039/P19960002029
PDF
The synthesis of lactam analogues of fentanyl
Ivan V. Miovi Goran M. Rogli M. D. Ivanovi Ljiljana Doen-Miovi Vesna D. Kiricojevi and Jelena B. Popovi
pg 2041; DOI:
10.1039/P19960002041
PDF
Lipase AKG mediated resolutions of ,-disubstituted 1,2-diols in organic solvents; remarkably high regio- and enantio-selectivity
Robert P. Hof and Richard M. Kellogg
pg 2051; DOI:
10.1039/P19960002051
PDF
From four-fold functionalised [3.3]cyclophanes to belt-shaped and multibridged molecules
Stefan Breidenbach Jörg Harren Susanne Neumann Martin Nieger Kari Rissanen and Fritz Vögtle
pg 2061; DOI:
10.1039/P19960002061
PDF
N-Halogeno compounds. Part 18. 1-Alkyl-4-fluoro-1,4-diazoniabicyclo[2.2.2]octane salts: user-friendly site-selective electrophilic fluorinating agents of the N-fluoroammonium class
R. Eric Banks Mohamed K. Besheesh Suad N. Mohialdin-Khaffaf and Iqbal Sharif
pg 2069; DOI:
10.1039/P19960002069
PDF
Corrigendum
Masaichi Naruse Sakae Aoyagi and Chihiro Kibayashi
pg 2077; DOI:
10.1039/P19960002077
PDF
Conference diary

pg xa; DOI:
10.1039/P199600000xa
PDF

Issue 17


Front cover

pg X069; DOI:
10.1039/P199600FX069
PDF
Back cover

pg X071; DOI:
10.1039/P199600BX071
PDF
Contents pages

pg P153; DOI:
10.1039/P199600FP153
PDF
Back matter

pg P159; DOI:
10.1039/P199600BP159
PDF
Biosynthesis of porphyrins and related macrocycles. Part 44. Synthetic and stereochemical studies on the proposed spiro intermediate for biosynthesis of the natural porphyrins
Mark A. Cassidy Nigel Crockett Finian J. Leeper and Alan R. Battersby
pg 2079; DOI:
10.1039/P19960002079
PDF
Biosynthesis of porphyrins and related macrocycles. Part 45. Determination by a novel X-ray method of the absolute configuration of the spiro lactam which inhibits uroporphyrinogen III synthase (cosynthetase)
Alan C. Spivey Alfredo Capretta Christopher S. Frampton Finian J. Leeper and Alan R. Battersby
pg 2091; DOI:
10.1039/P19960002091
PDF
A new procedure for the reduction of ,-unsaturated pyrrolidinones to 2H-pyrroles and 1H-pyrroles based on initial activation by N-nitrosation
Alan C. Spivey Christopher S. Frampton and Alan R. Battersby
pg 2103; DOI:
10.1039/P19960002103
PDF
Synthesis and absolute configurations of the naturally occurring 3- and 4-methylmuconolactones: X-ray structures of (S)-1-phenylethylammonium salts and an 8-bromo-1-methyl-muconodilactone
Andrew A. Freer Gordon W. Kirby Ghanakota V. Rao and Ronald B. Cain
pg 2111; DOI:
10.1039/P19960002111
PDF
Stereocontrolled route to some optically active -hydroxy phosphine oxides using the stereoselective addition of metallated phosphine oxides to proline-derived keto aminals
Peter O'Brien and Stuart Warren
pg 2117; DOI:
10.1039/P19960002117
PDF
Synthesis of (R)- or (S)-diphenylphosphinoyl hydroxy aldehydes and 1,2-diols using Mukaiyama's bicyclic aminal methodology and Sharpless asymmetric dihydroxylation
Peter O'Brien and Stuart Warren
pg 2129; DOI:
10.1039/P19960002129
PDF
Amino acids and peptides. Part 45. Development of a new N-protecting group of histidine, N-(1-adamantyloxymethyl)histidine, and its evaluation for peptide synthesis
Yoshio Okada Jidong Wang Takeshi Yamamoto Yu Mu and Toshio Yokoi
pg 2139; DOI:
10.1039/P19960002139
PDF
Coupling of ribofuranosyl fluoride and indoles
Masataka Yokoyama Mitsuru Nomura Hideo Togo and Hiroko Seki
pg 2145; DOI:
10.1039/P19960002145
PDF
Complex tetrahydrofurans from carbohydrate lactones: easy access to epimeric C-glycosides of glucofuranose from D-glycero-D-gulo-heptono-1,4-lactone
Claire J. F. Bichard Tilmann W. Brandstetter Juan C. Estevez George W. J. Fleet David J. Hughes and Joseph R. Wheatley
pg 2151; DOI:
10.1039/P19960002151
PDF
Novel method for the synthesis of - and -halogenonaphthalenes by regioselective benzannulation of aryl(gem-dihalogenocyclopropyl)methanols: application to the total synthesis of the lignan lactones, justicidin E and taiwanin C1
Yoo Tanabe Shinzo Seko Yoshinori Nishii Taichi Yoshida Naoka Utsumi and Gohfu Suzukamo
pg 2157; DOI:
10.1039/P19960002157
PDF
Molybdenum-mediated diastereoselective synthesis of 2-heterobicyclo[4.4.0]decene derivatives
Ming-Chang P. Yeh and Chong-Nan Chaung
pg 2167; DOI:
10.1039/P19960002167
PDF
Mechanism of arylation of nucleophiles by aryllead triacetates. Part 3. Concerning their reaction with phenols and X-ray molecular structure of p-methoxyphenyllead triacetate
Jacqueline Morgan Trevor W. Hambley and John T. Pinhey
pg 2173; DOI:
10.1039/P19960002173
PDF
New syntheses of 1-chloroalkylphosphinates
Xavier Morise Philippe Savignac and Jean-Marc Denis
pg 2179; DOI:
10.1039/P19960002179
PDF
Nucleophilic substitution of protected -bromoethyl cyclohexadiene-cis-diol as an alternative to direct microbial oxidation of -functionalized phenethyl substrates
Tomas Hudlicky Mary Ann A. Endoma and Gabor Butora
pg 2187; DOI:
10.1039/P19960002187
PDF
Podocarpane-to-spongian skeleton conversion. Synthesis of (+)-isoagatholactone and (–)-spongia-13(16),14-diene
Antonio Abad Consuelo Agulló Manuel Arnó M. Luisa Marín and Ramón J. Zaragozá
pg 2193; DOI:
10.1039/P19960002193
PDF
Regioselective alkylation of 2-phenylpyridines with terminal alkenes via C–H bond activation by a rhodium catalyst
Yeong-Gweon Lim Jung-Bu Kang and Yong Hae Kim
pg 2201; DOI:
10.1039/P19960002201
PDF
Rearrangement of methyl 11,12-di-O-methyl-6,7-didehydrocarnosate in basic medium. Easy hemisynthesis of miltirone
Javier G. Luis Lucía S. Andrés Winston Q. Fletcher El Hassane Lahlou and Aurea Perales
pg 2207; DOI:
10.1039/P19960002207
PDF
Pinacolization and reduction of aromatic carbonyls with aluminium–KOH
Jitender M. Khurana Arti Sehgal Amita Gogia (Late) Aparna Manian and Golak C. Maikap
pg 2213; DOI:
10.1039/P19960002213
PDF
Conference diary

pg viij; DOI:
10.1039/P1996000viij
PDF

Issue 18


Front cover

pg X073; DOI:
10.1039/P199600FX073
PDF
Back cover

pg X075; DOI:
10.1039/P199600BX075
PDF
Contents pages

pg P163; DOI:
10.1039/P199600FP163
PDF
Construction of the colchicine framework via two consecutive cyclopropane-mediated ring-expansion reactions
Martin G. Banwell Mariana Berak and David C. R. Hockless
pg 2217; DOI:
10.1039/P19960002217
PDF
Synthesis of 6-substituted pyrido[3,4-d]pyrimidin-4(3H)-ones via directed lithiation of 2-substituted 5-aminopyridine derivatives
Gordon W. Rewcastle William A. Denny R. Thomas Winters Norman L. Colbry and H. D. Hollis Showalter
pg 2221; DOI:
10.1039/P19960002221
PDF
Polar cycloaddition of 1-benzothiopyrylium salts with conjugated dienes and some transformations of the cycloadducts
Hiroshi Shimizu Shojiro Miyazaki and Tadashi Kataoka
pg 2227; DOI:
10.1039/P19960002227
PDF
Synthesis of 3,5-dithiothymidine and related compounds
Alessandra Eleuteri Colin B. Reese and Quanlai Song
pg 2237; DOI:
10.1039/P19960002237
PDF
Stereoselective isomerisations of 4-(3,5-dimethoxyphenyl)-2,5-dimethyl-1,3-dioxolanes. Temperature-dependent formation of either isochromanes or dihydroisobenzofurans
Robin G. F. Giles Rodney W. Rickards and Badra S. Senanayake
pg 2241; DOI:
10.1039/P19960002241
PDF
Novel cyclodehydration reaction of hydroxyphenols. An alternative to the Mitsunobu reaction
Panayiotis A. Procopiou Alastair C. Brodie Martyn J. Deal David F. Hayman and Gary M. Smith
pg 2249; DOI:
10.1039/P19960002249
PDF
6-Amino-1,8-dihydroimidazo[4,5-e][1,3]diazepin-4(5H)-one, a ring expanded analogue of guanine
Peter K. Bridson Huan Huang and Xiaoyan Lin
pg 2257; DOI:
10.1039/P19960002257
PDF
Reaction of carbanions generated from allylic phosphonates with -substituted cyclic enones
Malose J. Mphahlele and Tomasz A. Modro
pg 2261; DOI:
10.1039/P19960002261
PDF
Photochemical behaviour of -thiabicyclo[3.n.1]alkan-3-one: a mechanistic and exploratory study
Osamu Muraoka Bao-Zhong Zheng Maiko Nishimura and Genzoh Tanabe
pg 2265; DOI:
10.1039/P19960002265
PDF
Elemental fluorine. Part 6. Fluorination of cyclic 1,3-diketones and related compounds
Richard D. Chambers John Hutchinson Andrei S. Batsanov Christian W. Lehmann and Dimitrii Y. Naumov
pg 2271; DOI:
10.1039/P19960002271
PDF
Synthesis and nucleophilic properties of 1,2-dialkyl-3-nitropyrroles and 1,5-dialkyl-4-nitropyrrole-2-carboxylic acid derivatives
Antoni M. Molins-Pujol Concepció Moranta Carmina Arroyo M. Teresa Rodríguez M. Carmen Meca M. Dolors Pujol and Joaquim Bonal
pg 2277; DOI:
10.1039/P19960002277
PDF
Stereoselective synthesis of petrosterol and a formal synthesis of aragusterols
Toshio Honda Miho Katoh and Shin-ichi Yamane
pg 2291; DOI:
10.1039/P19960002291
PDF
Chiral dienes from enantiomerically pure enones. Highly stereoselective intramolecular Diels–Alder reaction involving ethenesulfonates
Guido Galley and Michael Pätzel
pg 2297; DOI:
10.1039/P19960002297
PDF
Synthesis and crystal structure determination of model compounds for the dibenzodioxocine structure occurring in wood lignins
Pirkko Karhunen Petteri Rummakko Aarne Pajunen and Gösta Brunow
pg 2303; DOI:
10.1039/P19960002303
PDF
Application of chemical P-450 model systems to studies on drug metabolism. Part X. Novel hydroxylactonization of ,- and ,- unsaturated carboxylic acids with an iron porphyrin–iodosylbenzene system
Masakatsu Komuro Tsunehiko Higuchi and Masaaki Hirobe
pg 2309; DOI:
10.1039/P19960002309
PDF
Novel linear polyene antibiotics: linearmycins
Shohei Sakuda Ursela Guce-Bigol Mutsuhiro Itoh Takashi Nishimura and Yasuhiro Yamada
pg 2315; DOI:
10.1039/P19960002315
PDF
An unprecedented cleavage of the -lactam ring: a novel synthesis of acyclic N,O- and N,S-acetals
Yasuyuki Kita Norio Shibata Noriyuki Kawano Naoki Yoshida Keita Matsumoto and Yasushi Takebe
pg 2321; DOI:
10.1039/P19960002321
PDF
Conference diary

pg xb; DOI:
10.1039/P199600000xb
PDF

Issue 19


Front cover

pg X077; DOI:
10.1039/P199600FX077
PDF
Back cover

pg X079; DOI:
10.1039/P199600BX079
PDF
Contents pages

pg P171; DOI:
10.1039/P199600FP171
PDF
Magnesiation of indoles with magnesium amide bases
Yoshinori Kondo Akihiro Yoshida and Takao Sakamoto
pg 2331; DOI:
10.1039/P19960002331
PDF
Unusual formation and X-ray crystal structure of stable anti-Bredt compounds by reaction of 3a,6a-diazapentalenes with dimethyl acetylenedicarboxylate
Kiyoshi Matsumoto Hirokazu Iida Hideki Katsura Takahisa Machiguchi Hidehiro Uekusa and Yuji Ohashi
pg 2333; DOI:
10.1039/P19960002333
PDF
Rhodium-catalysed decomposition of ,?-unsaturated -difluoro--diazo esters, the direct formation of bicyclo[2.1.0]pentane ring systems via intramolecular cyclopropanation
Guo-qiang Shi and Wei-ling Cai
pg 2337; DOI:
10.1039/P19960002337
PDF
Mechanistic aspects of the synthesis of 3-aminopyrroles from substituted 2-methyl-1,2-thiazolium salts or 3-aminothioacrylamides
Andreas Rolfs Peter G. Jones and Jürgen Liebscher
pg 2339; DOI:
10.1039/P19960002339
PDF
Studies on pyrazines. Part 32. Synthesis of trisubstituted and tetrasubstituted pyrazines as ant pheromones
Nobuhiro Sato and Tomoyuki Matsuura
pg 2345; DOI:
10.1039/P19960002345
PDF
Reaction of 2-amino- and 2-(substituted amino)-1-azaazulenes with chloro-, phenyl- and diphenyl-ketene
Noritaka Abe Ichiro Osaki Sawako Kojima Haruhiko Matsuda Yoshikazu Sugihara and Akikazu Kakehi
pg 2351; DOI:
10.1039/P19960002351
PDF
Biosynthesis of ML-236C and the hypocholesterolemic agents compactin by Penicillium aurantiogriseum and lovastatin by Aspergillus terreus: determination of the origin of carbon, hydrogen and oxygen atoms by 13C NMR spectrometry and observation of unusual labelling of acetate-derived oxygens by 18O2
Kurt Wagschal Yuko Yoshizawa David J. Witter Yaoquan Liu and John C. Vederas
pg 2357; DOI:
10.1039/P19960002357
PDF
Convenient route for the synthesis of 3-substituted and 3,4-disubstituted pyrrole-2,5-dicarbaldehydes
Silvano Cadamuro Iacopo Degani Rita Fochi Antonella Gatti and Laura Piscopo
pg 2365; DOI:
10.1039/P19960002365
PDF
Comparison of the substrate specificity of type I and type II dehydroquinases with 5-deoxy- and 4,5-dideoxy-dehydroquinic acid
Joanna M. Harris William J. Watkins Alastair R. Hawkins John R. Coggins and Chris Abell
pg 2371; DOI:
10.1039/P19960002371
PDF
Tirucalla-5,24-dien-3-ol [(13,14,17,20S)-lanosta-5,24-dien-3-ol] and three other 5-unsaturated tirucallanes from the roots of Bryonia dioica Jacq.: the first naturally occurring C-10 methylated tetracyclic triterpene alcohols with a 5-monounsaturated skeleton
Toshihiro Akihisa Yumiko Kimura Wilhelmus C. M. C. Kokke Sei-ichi Takase Ken Yasukawa and Toshitake Tamura
pg 2379; DOI:
10.1039/P19960002379
PDF
Iron(III)-catalysed nitration of non-activated and moderately activated arenes with nitrogen dioxide–molecular oxygen under neutral conditions
Hitomi Suzuki Shuji Yonezawa Nobuaki Nonoyama and Tadashi Mori
pg 2385; DOI:
10.1039/P19960002385
PDF
Synthesis of 1- and 2-substituted thianthrenes
James M. Lovell and John A. Joule
pg 2391; DOI:
10.1039/P19960002391
PDF
Reactions of endocyclic linearly conjugated dienolates with Michael acceptors leading to bicyclo[2.2.2]octane derivatives. Application to the synthesis of C13 degradation products of carotenoids
Nobuhiko Ito and Takeaki Etoh
pg 2397; DOI:
10.1039/P19960002397
PDF
Synthesis and some properties of mixed alkyldi-(–)-menthyltin hydrides
Cristian A. Vitale and Julio C. Podestá
pg 2407; DOI:
10.1039/P19960002407
PDF
Synthesis of the cyclic heptapeptides axinastatin 2 and axinastatin 3
George R. Pettit Jeffrey W. Holman and Gerard M. Boland
pg 2411; DOI:
10.1039/P19960002411
PDF
Conference diary

pg viik; DOI:
10.1039/P1996000viik
PDF

Issue 20


Front cover

pg X081; DOI:
10.1039/P199600FX081
PDF
Back cover

pg X083; DOI:
10.1039/P199600BX083
PDF
Contents pages

pg P177; DOI:
10.1039/P199600FP177
PDF
Back matter

pg P185; DOI:
10.1039/P199600BP185
PDF
Palladium-catalysed hydrostannylations of 1-bromoalkynes. A practical synthesis of (E)-1-stannylalk-1-enes
Christopher D. J. Boden Gerald Pattenden and Tao Ye
pg 2417; DOI:
10.1039/P19960002417
PDF
Porphyrin–cholic acid–chlorambucil triads: synthesis and light-induced nuclease activity
Goverdhan Mehta Sengodagounder Muthusamy Bhaskar G. Maiya and Mallena Sirish
pg 2421; DOI:
10.1039/P19960002421
PDF
Approaches to synthetic neolignans
Kaichang Li and Richard F. Helm
pg 2425; DOI:
10.1039/P19960002425
PDF
Indole-fused tetraazacyclooctadecanes: double-helical macrocycles
Mark Mascal Ian G. Wood Michael J. Begley Andre S. Batsanov Timothy Walsgrove Alexandra M. Z. Slawin David J. Williams Alex F. Drake and Giuliano Siligardi
pg 2427; DOI:
10.1039/P19960002427
PDF
Directed evolution of trypsin inhibiting peptides using a genetic algorithm
Yohei Yokobayashi Kazunori Ikebukuro Scott McNiven and Isao Karube
pg 2435; DOI:
10.1039/P19960002435
PDF
Heterocyclic -hydroxy--amino acids as substrates for a novel aldolase from Streptomyces amakusaensis; preparation of (2R,3R)-3-(2-thienyl)serine and (2R,3R)-3-(2-furyl)serine from racemic threo material
Matthew Bycroft Richard B. Herbert and George J. Ellames
pg 2439; DOI:
10.1039/P19960002439
PDF
Synthesis of some substituted quinoxalines and polycyclic systems containing the quinoxaline nucleus
Abid R. Ahmad Lina K. Mehta and John Parrick
pg 2443; DOI:
10.1039/P19960002443
PDF
New -electron donor systems based on acenaphtho[1,2-b][1,4]dithiine
Martin R. Bryce Antony Chesney Alexander K. Lay Andrei S. Batsanov and Judith A. K. Howard
pg 2451; DOI:
10.1039/P19960002451
PDF
Approaches to the stepwise synthesis of benzoporphyrins and phthalocyanines. Part 1. Synthesis of opp-dibenzoporphyrins (dibenzo[g,q]porphyrins)
Raymond Bonnett and Kimberly A. McManus
pg 2461; DOI:
10.1039/P19960002461
PDF
Asymmetric synthesis of (R)-hexane-1,5-diol, (R)-hex-3-ene-1,5-diol and (R)-6-methylhept-5-en-2-ol (sulcatol) employing a tandem asymmetric conjugate addition and stereospecific Meisenheimer rearrangement protocol
Stephen G. Davies and G. Darren Smyth
pg 2467; DOI:
10.1039/P19960002467
PDF
Chymotrypsin inhibitory conformation induced by amino acid side chain–side chain intramolecular CH/ interaction
Yasuyuki Shimohigashi Iori Maeda Takeru Nose Koichi Ikesue Hiroshi Sakamoto Tomohisa Ogawa Yuzuru Ide Megumi Kawahara Takashi Nezu Yoshihiro Terada Keiichi Kawano and Motonori Ohno
pg 2479; DOI:
10.1039/P19960002479
PDF
Diastereoselective hydrogenations of -alkyl -(2,3,4,6-tetra-O-acetyl--D-glucopyranosyloxy)methylene carbonyl compounds. New route to stereopure -alkyl -oxymethyl carbonyl compounds
David S. Larsen Anthony Schofield Richard J. Stoodley and Peter D. Tiffin
pg 2487; DOI:
10.1039/P19960002487
PDF
Total synthesis of the -adrenergic receptor antagonist, the tetrahydroisoquinoline MY336-a and its epimer
Teodoro S. Kaufman
pg 2497; DOI:
10.1039/P19960002497
PDF
Acid-catalysed rearrangement of caryophyllene oxide
Wing-Yan Tsui and Geoffrey Brown
pg 2507; DOI:
10.1039/P19960002507
PDF
A new entry to the synthesis of 5-substituted 1,2,3-triazines by reaction with silyl enol ethers and ceric ammonium nitrate
Takashi Itoh Yûji Matsuya Hiroshi Hasegawa Kazuhiro Nagata Mamiko Okada and Akio Ohsawa
pg 2511; DOI:
10.1039/P19960002511
PDF
Reactivity of perfluoro-(cis-2,3-dialkyloxaziridines) with heteroaromatic nitrogen compounds
Rosanna Bernardi Barbara Novo and Giuseppe Resnati
pg 2517; DOI:
10.1039/P19960002517
PDF
Transannular cyclization reactions of cyclooctane-1,5-dione and 5-ethoxycarbonylmethylenecyclooctanone upon treatment with diamines. An efficient one-pot synthesis of substituted 2,6-diazatricyclo[5.3.3.01,6]- and 2,5-diazatricyclo[4.3.3.01,5]-alkanes and a study of their acetylation products
Elizabeth Malamidou-Xenikaki
pg 2523; DOI:
10.1039/P19960002523
PDF
Stereoselective synthesis of trifluoromethylated -chloro-,-unsaturated esters and nitriles
Yanchang Shen and Shu Gao
pg 2531; DOI:
10.1039/P19960002531
PDF
Absolute configuration of flavanone–benzofuranone-type biflavonoids and 2-benzyl-2-hydroxybenzofuranones
Riaan Bekker E. Vincent Brandt and Daneel Ferreira
pg 2535; DOI:
10.1039/P19960002535
PDF
Reactivity of 3-benzylidene- and 3-ethylidene-2,3-dihydro-2-methyl-1,2-benzothiazin-4-one 1,1-dioxide towards alkylidenephosphoranes
Piero Dalla Croce and Concetta La Rosa
pg 2541; DOI:
10.1039/P19960002541
PDF
Reductive alkylation of pyridinium salts. Part 1. Synthesis of di-, tetra- and hexa-hydropyridine esters
John MacTavish George R. Proctor and James Redpath
pg 2545; DOI:
10.1039/P19960002545
PDF
Reductive alkylation of pyridinium salts. Part 2. Utilisation of di-, tetra- and hexa-hydropyridine esters
Kevin J. McCullough John MacTavish George R. Proctor and James Redpath
pg 2553; DOI:
10.1039/P19960002553
PDF
Conference diary

pg xc; DOI:
10.1039/P199600000xc
PDF

Issue 21


Front cover

pg X085; DOI:
10.1039/P199600FX085
PDF
Advertisements

pg X087; DOI:
10.1039/P1996000X087
PDF
Back cover

pg X091; DOI:
10.1039/P199600BX091
PDF
Contents pages

pg P187; DOI:
10.1039/P199600FP187
PDF
New entry to benzo[b]thieno[2,3-b]- and benzo[b]thieno-[3,2-b]-pyridines using 2- and 3-azidobenzo[b]thiophene as the nitrogen precursors
Alessandro Degl'Innocenti Maria Funicello Patrizia Scafato Piero Spagnolo and Paolo Zanirato
pg 2561; DOI:
10.1039/P19960002561
PDF
Chemoenzymatic routes to chiral (non-racemic) cyclopropanes. Preparation of a key intermediate for the synthesis of (1R)-cis-pyrethroids
Martin G. Banwell and Grant S. Forman
pg 2565; DOI:
10.1039/P19960002565
PDF
Investigation of the configurational stability of lithiated phosphine oxides using diastereomerically pure and enantiomerically enriched phosphine oxides
Peter O'Brien and Stuart Warren
pg 2567; DOI:
10.1039/P19960002567
PDF
A reactivity study of [6-(tert-butylsulfonyl)benzene]-tricarbonylchromium(0)
Susan E. Gibson (née Thomas) Nathalie Guillo Andrew J. P. White and David J. Williams
pg 2575; DOI:
10.1039/P19960002575
PDF
Synthesis of sibutramine, a novel cyclobutylalkylamine useful in the treatment of obesity, and its major human metabolites
James E. Jeffery Frank Kerrigan Thomas K. Miller Graham J. Smith and Gerald B. Tometzki
pg 2583; DOI:
10.1039/P19960002583
PDF
Synthesis of neoflavones by Suzuki arylation of 4-substituted coumarins
Gerard M. Boland Dervilla M. X. Donnelly Jean-Pierre Finet and Martin D. Rea
pg 2591; DOI:
10.1039/P19960002591
PDF
Formation of 1,2,3,4-dibenzocycl[2.2.3]azines by a novel consecutive 1,3-dipolar cycloaddition of pyridinium dicyanomethylides to benzyne
Kiyoshi Matsumoto Hideki Katsura Takane Uchida Kinuyo Aoyama and Takahisa Machiguchi
pg 2599; DOI:
10.1039/P19960002599
PDF
Radical-mediated cyclisation of -aryl--dicarbonyl compounds to -tetralones [3,4-dihydronaphthalen-2(1H)-ones]
Joanne F. Jamie and Rodney W. Rickards
pg 2603; DOI:
10.1039/P19960002603
PDF
Quinones. Part 14. Attempted synthesis of 9,10-dimethyl-2,6-anthraquinone. Desmotropic formation of secondary ortho-anthraquinoles instead of 1,2-anthrahydroquinones
Peter Boldt Stephan Zippel and Michael Ratzkowsky
pg 2615; DOI:
10.1039/P19960002615
PDF
Enantiodivergent synthesis of both enantiomers of the macrocyclic lactone lasiodiplodin
Franz Bracher and Brigitte Schulte
pg 2619; DOI:
10.1039/P19960002619
PDF
Characterization of lanthanide-mediated DNA cleavage by intercalator-linked hydroxamic acids: comparison with transition systems
Shigeki Hashimoto and Yushin Nakamura
pg 2623; DOI:
10.1039/P19960002623
PDF
Preparation of 14-nitrocamptothecin derivatives by reactions of camptothecin with nitronium tetrafluoroborate in acidic solvents
Zhisong Cao
pg 2629; DOI:
10.1039/P19960002629
PDF
Synthesis of analogues of porphobilinogen
Finian J. Leeper Martin Rock and Diana Appleton
pg 2633; DOI:
10.1039/P19960002633
PDF
Interaction of analogues of porphobilinogen with porphobilinogen deaminase
Finian J. Leeper and Martin Rock
pg 2643; DOI:
10.1039/P19960002643
PDF
Preparative transformation of natural phospholipids catalysed by phospholipase D from Streptomyces
Paola D'Arrigo Lorenzo de Ferra Valentino Piergianni Antonio Selva Stefano Servi and Alberto Strini
pg 2651; DOI:
10.1039/P19960002651
PDF
Enzyme-mediated synthesis of two diastereoisomeric forms of phosphatidylglycerol and of diphosphatidylglycerol (cardiolipin)
Paola D'Arrigo Lorenzo de Ferra Giuseppe Pedrocchi-Fantoni Domenico Scarcelli Stefano Servi and Alberto Strini
pg 2657; DOI:
10.1039/P19960002657
PDF
Corrigenda
Richard F. W. Jackson Andrew D. Briggs Paul A. Brown William Clegg Mark R. J. Elsegood Christopher Frampton Robert S. Atkinson and Paul J. Williams
pg 2661; DOI:
10.1039/P19960002661
PDF
Conference diary

pg viil; DOI:
10.1039/P1996000viil
PDF

Issue 22


Front cover

pg X093; DOI:
10.1039/P199600FX093
PDF
Back cover

pg X095; DOI:
10.1039/P199600BX095
PDF
Contents pages

pg P193; DOI:
10.1039/P199600FP193
PDF
Cross-coupling reaction of cyclopropylboronic acid with bromoarenes
Xiang-Zhu Wang and Ming-Zhi Deng
pg 2663; DOI:
10.1039/P19960002663
PDF
-Face selectivities in nucleophilic additions to 2-endo-arylnorbornan-7-ones: the role of through-space electrostatic interactions
Goverdhan Mehta Faiz Ahmed Khan Narinder Mohal I. N. Narayan Namboothiri P. Kalyanaraman and Jayaraman Chandrasekhar
pg 2665; DOI:
10.1039/P19960002665
PDF
Synthesis of a chiral azodicarboxamide containing a bridging binaphthyl moiety: electrophilic amination reactions of achiral ester enolates
Joanna M. Harris Robert McDonald and John C. Vederas
pg 2669; DOI:
10.1039/P19960002669
PDF
Investigation of a reverse approach to extended porphyrin systems. Synthesis of a 2,3-diaminoporphyrin and its reactions with -diones
Maxwell J. Crossley Lionel G. King Ian A. Newsom and Craig S. Sheehan
pg 2675; DOI:
10.1039/P19960002675
PDF
Synthesis of a series of trifluoromethylazoles and determination of pKa of acidic and basic trifluoromethyl heterocycles by 19F NMR spectroscopy
Brian G. Jones Sarah K. Branch Andrew S. Thompson and Michael D. Threadgill
pg 2685; DOI:
10.1039/P19960002685
PDF
Synthesis of sulfoxides by the oxidation of sulfides with sodium chlorite catalysed by manganese(III) acetylacetonate in acetone in the presence of alumina
Masao Hirano Shigetaka Yakabe James H. Clark and Takashi Morimoto
pg 2693; DOI:
10.1039/P19960002693
PDF
Syntheses of 1-substituted furan-fused 3-sulfolenes and their Diels–Alder reactions
Takayoshi Suzuki Hideyuki Fuchii and Hiroaki Takayama
pg 2699; DOI:
10.1039/P19960002699
PDF
Magnesium methoxide complexation in the control of chemical reactions
S. Richard Baker Michael L. F. Cadman Leslie Crombie David A. V. Edwards and Jayshree Mistry
pg 2705; DOI:
10.1039/P19960002705
PDF
Reactions of fused and unfused -pyrones with magnesium alkoxide, sodium alkoxide and water as the nucleophile: effects of chelation
Leslie Crombie David E. Games and Alun W. G. James
pg 2715; DOI:
10.1039/P19960002715
PDF
Aziridination of N-sulfonylimines with a stabilized sulfonium ylide: simple preparation of N-sulfonyl-2-[(E)-2-(alkoxycarbonyl)ethenyl]-3-arylaziridines
An-Hu Li Li-Xin Dai and Xue-Long Hou
pg 2725; DOI:
10.1039/P19960002725
PDF
Preparation of selenoxides from the catalytic autoxidation of organoselenides with nitrogen oxides
Eric Bosch and Jay K. Kochi
pg 2731; DOI:
10.1039/P19960002731
PDF
Preparation of carbocyclic analogues of 2-deoxyribonucleotides possessing a phosphonate substituent at the 5-position
Alex F. Drake Antonio Garofalo Jennifer M. L. Hillman Valeria Merlo Ray McCague and Stanley M. Roberts
pg 2739; DOI:
10.1039/P19960002739
PDF
A highly stereoselective synthesis of 3-hydroxy-1-aryltetralin lignans based on the stereoselective hydroxylation of ,-dibenzyl--butyro-lactones: the first synthesis of ()-cycloolivil
Yasunori Moritani Tatsuzo Ukita Hajime Hiramatsu Kimio Okamura Hiroshi Ohmizu and Tameo Iwasaki
pg 2747; DOI:
10.1039/P19960002747
PDF
Synthesis, conformation and tropicity of dimethano-bridged tetradehydrothia[21]-, -[23]- and -[25]annulenes
Jro Ojima Naoki Hiraiwa Hiroyuki Higuchi Ikuko Kobayashi Koji Yamamoto Toshikatsu Yoshida Tomohiro Adachi Hiroshi Matsubara and Gaku Yamamoto
pg 2755; DOI:
10.1039/P19960002755
PDF
Synthesis of 16-[carbamoyl(bromomethyl)alkyl]estradiol: a potential dual-action inhibitor designed to blockade estrogen action and biosynthesis
Martin R. Tremblay and Donald Poirier
pg 2765; DOI:
10.1039/P19960002765
PDF
Conference diary

pg viim; DOI:
10.1039/P1996000viim
PDF

Issue 23


Front cover

pg X097; DOI:
10.1039/P199600FX097
PDF
Back cover

pg X099; DOI:
10.1039/P199600BX099
PDF
Contents pages

pg P199; DOI:
10.1039/P199600FP199
PDF
Generation and trapping of 1,3-dithian-2-ylidene-substituted ethyl carbene. On the existence of 4,8-dithiaspiro[2.5]oct-1-ene
Hans-Georg Schwarz and Ernst Schaumann
pg 2773; DOI:
10.1039/P19960002773
PDF
Lipase-catalysed esterification of some -D-glucopyranosides in dry media under focused microwave irradiation
Mirjana Gelo-Pujic Eryka Guibé-Jampel André Loupy Saskia A. Galema and Daniel Mathé
pg 2777; DOI:
10.1039/P19960002777
PDF
Enthalpic (electrostatic) contribution to the chelate effect: a correlation between ligand binding constant and a specific hydrogen bond strength in complexes of glycopeptide antibiotics with cell wall analogues
Mark S. Searle Gary J. Sharman Patrick Groves Bellinda Benhamu Daniel A. Beauregard Martin S. Westwell Robert J. Dancer Alison J. Maguire Andrew C. Try and Dudley H. Williams
pg 2781; DOI:
10.1039/P19960002781
PDF
Isatin chloride: a phantom. Reactions of 2-(2,2-dichloro-2,3-dihydro-3-oxoindol-1-yl)-3H-indol-3-one
Sir John Cornforth Peter B. Hitchcock and Panteleimon Rozos
pg 2787; DOI:
10.1039/P19960002787
PDF
Effects of catalysts on the cyclization of 2-diazo-2-methoxycarbonyl-N-aryl-N-alkylethanamides
Keith Smith and Dawoud Bahzad
pg 2793; DOI:
10.1039/P19960002793
PDF
Domino syntheses of five-, six- and seven-membered O-, N- and S-heterocycles from -, - and -substituted carboxylic esters
J. Löffler and R. Schobert
pg 2799; DOI:
10.1039/P19960002799
PDF
Chemistry of silyl thioketones. Part 10. Synthesis and reactivity of -silyl vinyl sulfides
Bianca Flavia Bonini Mauro Comes-Franchini Mariafrancesca Fochi Germana Mazzanti Francesca Peri and Alfredo Ricci
pg 2803; DOI:
10.1039/P19960002803
PDF
Synthesis and biological evaluation of sulfur isosters of the potent influenza virus sialidase inhibitors 4-amino-4-deoxy- and 4-deoxy-4-guanidino-Neu5Ac2en
Gaik B. Kok Michael Campbell Brendan Mackey and Mark von Itzstein
pg 2811; DOI:
10.1039/P19960002811
PDF
Synthesis of C-4-disubstituted analogues of N-acetylneuraminic acid
Darrin R. Groves and Mark Von Itzstein
pg 2817; DOI:
10.1039/P19960002817
PDF
Asymmetric titanium-catalysed Michael addition of O-benzylhydroxylamine to -unsaturated carbonyl compounds: synthesis of -amino acid precursors
Lise Falborg and Karl Anker Jørgensen
pg 2823; DOI:
10.1039/P19960002823
PDF
Ambient temperature method for the generation and Diels–Alder trapping of benzofuran-2,3-quinodimethane (2,3-dimethylidene-2,3-dihydrobenzofuran)
Simon B. Bedford (the late) Michael J. Begley Philip Cornwall Joel P. Foreman and David W. Knight
pg 2827; DOI:
10.1039/P19960002827
PDF
Synthesis of cleviolide and the scobinolides
Gregory J. Hollingworth Alexandre M. E. Richecoeur and Joseph Sweeney
pg 2833; DOI:
10.1039/P19960002833
PDF
Development of the Juli asymmetric epoxidation reaction. Part 2. Application of the oxidation to alkyl enones, enediones and unsaturated keto esters
Wolfgang Kroutil M. Elena Lasterra-Sánchez Samuel J. Maddrell Patrick Mayon Phillip Morgan Stanley M. Roberts Steven R. Thornton Christine J. Todd and Melek Tüter
pg 2837; DOI:
10.1039/P19960002837
PDF
Convenient synthesis of (2R)- and (2S)-2-(1-methylethyl)-5-oxo-2-phenylpentanenitrile, intermediates in the preparation of phenylalkylamine calcium channel blockers
Jeremy Gilmore Will Prowse David Steggles Michael Urquhart and Jennifer Olkowski
pg 2845; DOI:
10.1039/P19960002845
PDF
Efficient synthesis of 1-methylcarbapenems based on the counter-attack strategy
Masahiko Seki Kazuhiko Kondo and Tameo Iwasaki
pg 2851; DOI:
10.1039/P19960002851
PDF
New route to 4-alkoxyquinazoline-2-carbonitriles
Thierry Besson and Charles W. Rees
pg 2857; DOI:
10.1039/P19960002857
PDF
Effective transgalactosylation catalysed by a lipid-coated -D-galactosidase in organic solvents
Yoshio Okahata and Toshiaki Mori
pg 2861; DOI:
10.1039/P19960002861
PDF
Conference diary

pg viin; DOI:
10.1039/P1996000viin
PDF

Issue 24


Front cover

pg X101; DOI:
10.1039/P199600FX101
PDF
Back cover

pg X103; DOI:
10.1039/P199600BX103
PDF
Contents pages

pg P205; DOI:
10.1039/P199600FP205
PDF
-Chymotrypsin-catalysed peptide synthesis using activated esters as acyl donors
Toshifumi Miyazawa Shin'ichi Nakajo Miyako Nishikawa Kiwamu Imagawa Ryoji Yanagihara and Takashi Yamada
pg 2867; DOI:
10.1039/P19960002867
PDF
Effective enantioselective approach to -aminoalkylacrylic acid derivatives via a synthetic equivalent of an asymmetric Baylis–Hillman reaction: application to the synthesis of two C-2 hydroxymethyl analogues of docetaxel
Yves Génisson Christine Massardier Isabelle Gautier-Luneau and Andrew E. Greene
pg 2869; DOI:
10.1039/P19960002869
PDF
Reliable method for the synthesis of aryl -D-glucopyranosides, using boron trifluoride–diethyl ether as catalyst
Elly Smits Jan B. F. N. Engberts Richard M. Kellogg and Henk A. van Doren
pg 2873; DOI:
10.1039/P19960002873
PDF
N–H insertion reactions of rhodium carbenoids. Part 1. Preparation of -amino acid and -aminophosphonic acid derivatives
Enrique Aller Richard T. Buck Martin J. Drysdale Leigh Ferris David Haigh Christopher J. Moody Neil D. Pearson and J. Bobby Sanghera
pg 2879; DOI:
10.1039/P19960002879
PDF
N–H insertion reactions of rhodium carbenoids. Part 2. Preparation of N-substituted amino(phosphoryl)acetates (N-substituted phosphorylglycine esters)
Leigh Ferris David Haigh and Christopher J. Moody
pg 2885; DOI:
10.1039/P19960002885
PDF
Synthesis of substituted dibenzophospholes. Part 9. Preparation of two water-soluble phosphinic–polyphosphonic acids
Sir John Cornforth
pg 2889; DOI:
10.1039/P19960002889
PDF
Anomalous fluorinations of 3-aryl-2-hydroxypropanoic esters by diethylaminosulfur trifluoride (DAST)
David Haigh Lee J. Jefcott Katherine Magee and Hamish McNab
pg 2895; DOI:
10.1039/P19960002895
PDF
Catalytic enantioselective reaction. Part 9. 1,2-O-Isopropylidene-5-deoxy-5-N,N-dialkyl (or -N-monoalkyl)amino--D-xylofuranose derivatives as highly effective chiral catalysts for enantioselective addition of diethylzinc to aliphatic and aromatic aldehydes
Byung Tae Cho and Namdu Kim
pg 2901; DOI:
10.1039/P19960002901
PDF
Reactions of 2-methyl-3,1-benzoxazin-4-one with active methylene compounds: a new route to 3-substituted 4-hydroxyquinolin-2(1H)-ones
Anastasia Detsi Vassilios Bardakos John Markopoulos and Olga Igglessi-Markopoulou
pg 2909; DOI:
10.1039/P19960002909
PDF
Occurrence of phenylpyruvic acid in woody plants: biosynthetic significance and synthesis of an enolic glucoside derivative
Charlene Marais Jacobus A. Steenkamp and Daneel Ferreira
pg 2915; DOI:
10.1039/P19960002915
PDF
[1,4] and [2,3] Sigmatropic rearrangements of ylides generated from N-(-cyano)allyl-N-cyanomethyl-N,N-dimethylammonium perchlorates
Andrzej Joczyk Tadeusz Zdrojewski Pawe Grzywaca and Pawe Balcerzak
pg 2919; DOI:
10.1039/P19960002919
PDF
Syntheses of piperidine and perhydroazepine derivatives, precursors of two selective antagonists of muscarinic M2 receptors: AF-DX 384 and its perhydroazepine isomer
Cécile Perrio-Huard Christophe Ducandas Marie Claire Lasne and Bernard Moreau
pg 2925; DOI:
10.1039/P19960002925
PDF
Analysis of the reactivity of the dithioacetal mono-S-oxide 1-deoxy-1-ethylsulfinyl-1-ethylthio-3,4-O-isopropylidene-D-erythritol under different conditions of reduction
Yolanda Arroyo-Gómez Juan A. López-Sastre J. Felix Rodríguez-Amo and Ma Ascension Sanz-Tejedor
pg 2933; DOI:
10.1039/P19960002933
PDF
Helical thiaza[2.2]metacyclophanes. Synthesis, structure, circular dichroism, absolute configuration
Dirk Müller Marc Böhme Martin Nieger Kari Rissanen and Fritz Vögtle
pg 2937; DOI:
10.1039/P19960002937
PDF
Conference diary

pg xv; DOI:
10.1039/P199600000xv
PDF